EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.1.1.1 | 0.06 |
- |
N1-methylnicotinamide |
IC50 0.06 mM for human protein, 0.03 mM for recombinant protein |
441255 |
2.1.1.1 | 0.0012 |
- |
S-adenosyl-L-homocysteine |
substrate S-adenosyl-L-methionine, pH 8.6, 37°C |
756053 |
2.1.1.1 | 0.002 |
- |
S-adenosyl-L-homocysteine |
substrate quinoline, pH 8.6, 37°C |
756053 |
2.1.1.1 | 0.023 |
- |
1-methylnicotinamide |
substrate quinoline, pH 8.6, 37°C |
756053 |
2.1.1.1 | 0.000588 |
- |
6-(methylamino)pyridine-3-carboxamide |
pH 7.5, 37°C |
756192 |
2.1.1.1 | 0.000837 |
- |
6-methoxy-4-methylpyridine-3-carboxamide |
pH 7.5, 37°C |
756192 |
2.1.1.1 | 0.0012 |
- |
3-amino-6-fluoro-1-methylquinolin-1-ium |
pH 8.6, 37°C |
757392 |
2.1.1.1 | 0.0012 |
- |
5-amino-1-methylquinolin-1-ium |
pH 8.6, 37°C |
757392 |
2.1.1.1 | 0.0018 |
- |
1,8-dimethylquinolin-1-ium |
pH 8.6, 37°C |
757392 |
2.1.1.1 | 0.0026 |
- |
7-amino-1-methylquinolin-1-ium |
pH 8.6, 37°C |
757392 |