EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.6.5.5 | 0.0051 |
- |
(5Z)-5-[(6,8-dichloro-4-oxo-4H-chromen-3-yl)methylidene]-3-ethyl-2-thioxo-1,3-thiazolidin-4-one |
pH and temperature not specified in the publication |
718468 |
3.6.5.5 | 0.0051 |
- |
2-cyano-N-[3-[2-cyano-3-(3,4-dihydroxyphenyl)acryloylamino]-2-hydroxypropyl]-3-(3,4-dihydroxyphenyl)acrylamide |
IC50: 0.0051 mM |
669796 |
3.6.5.5 | 0.0051 |
- |
catechol-acrylamide |
IC50: 0.0051 mM |
669796 |
3.6.5.5 | 0.0055 |
- |
(5Z)-5-[(5-chloro-1-benzothiophen-3-yl)methylidene]-2-thioxo-1,3-thiazolidin-4-one |
pH and temperature not specified in the publication |
718468 |
3.6.5.5 | 0.0055 |
- |
[(5Z)-5-(3,5-dichlorobenzylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]acetic acid |
pH and temperature not specified in the publication |
718468 |
3.6.5.5 | 0.006 |
- |
2-cyano-N-[3-[2-cyano-3-(3,4,5-trihydroxyphenyl)acryloylamino]hexyl]-3-(3,4,5-trihydroxyphenyl)acrylamide |
IC50: 0.006 mM |
669796 |
3.6.5.5 | 0.0064 |
- |
3-(4-azidophenyl)-2-cyano-N-[3-[2-cyano-3-(3,4-dihydroxyphenyl)acryloylamino]propyl]acrylamide |
in 10 mM Tris, 10 mM NaCl, 2 mM Mg2+, at 30°C |
697337 |
3.6.5.5 | 0.0068 |
- |
4-(N,N-dimethyl-N-dodecyl-N-propyl)-4-aza-10-oxa-6-ethyltricyclo[5.2.1]decane-3,5-dione methanesulfonate |
- |
689237 |
3.6.5.5 | 0.0071 |
- |
(5Z)-5-[4-[3-(dimethylamino)propoxy]benzylidene]-3-ethyl-2-thioxo-1,3-thiazolidin-4-one |
pH and temperature not specified in the publication |
718468 |
3.6.5.5 | 0.0073 |
- |
sertraline |
in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C |
696551 |