3.6.5.5 additional information - additional information IC50 values, overview 757390 3.6.5.5 0.0017 - 2-cyano-N-[2-[2-cyano-3-(3,4,5-trihydroxyphenyl)acryloylamino]ethyl]-3-(3,4,5-trihydroxyphenyl)acrylamide IC50: 0.0017 mM 669796 3.6.5.5 0.0017 - bis-tyrphostin in 10 mM Tris, 10 mM NaCl, 2 mM Mg2+, at 30°C 697337 3.6.5.5 0.0023 - 4-(N,N-dimethyl-N-octadecyl-N-ethyl)-4-aza-10-oxatricyclo[5.2.1]decane-3,5-dione bromide - 689237 3.6.5.5 0.0031 - (5Z)-5-(3,5-dichlorobenzylidene)-3-ethyl-2-thioxo-1,3-thiazolidin-4-one pH and temperature not specified in the publication 718468 3.6.5.5 0.0034 - [(5Z)-5-[(6,8-dichloro-4-oxo-4H-chromen-3-yl)methylidene]-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]acetic acid pH and temperature not specified in the publication 718468 3.6.5.5 0.0044 - 3-[(5Z)-5-(3,5-dichlorobenzylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]propanoic acid pH and temperature not specified in the publication 718468 3.6.5.5 0.0045 - (5Z)-5-[4-[3-(dimethylamino)propoxy]benzylidene]-3-(prop-2-en-1-yl)-2-thioxo-1,3-thiazolidin-4-one pH and temperature not specified in the publication 718468 3.6.5.5 0.005 - 2-cyano-N-[3-[2-cyano-3-(3,4-dihydroxy-5-methoxyphenyl)acryloylamino]propyl]-3-(3,4-dihydroxy-5-meth-oxyphenyl)acrylamide IC50: 0.005 mM 669796 3.6.5.5 0.0051 - (2E,2'E)-N,N'-(2-hydroxypropane-1,3-diyl)bis[2-cyano-3-(3,4-dihydroxyphenyl)prop-2-enamide] in 10 mM Tris, 10 mM NaCl, 2 mM Mg2, at 30°C 697337 3.6.5.5 0.0051 - (5Z)-5-[(6,8-dichloro-4-oxo-4H-chromen-3-yl)methylidene]-3-ethyl-2-thioxo-1,3-thiazolidin-4-one pH and temperature not specified in the publication 718468 3.6.5.5 0.0051 - 2-cyano-N-[3-[2-cyano-3-(3,4-dihydroxyphenyl)acryloylamino]-2-hydroxypropyl]-3-(3,4-dihydroxyphenyl)acrylamide IC50: 0.0051 mM 669796 3.6.5.5 0.0051 - catechol-acrylamide IC50: 0.0051 mM 669796 3.6.5.5 0.0055 - (5Z)-5-[(5-chloro-1-benzothiophen-3-yl)methylidene]-2-thioxo-1,3-thiazolidin-4-one pH and temperature not specified in the publication 718468 3.6.5.5 0.0055 - [(5Z)-5-(3,5-dichlorobenzylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]acetic acid pH and temperature not specified in the publication 718468 3.6.5.5 0.006 - 2-cyano-N-[3-[2-cyano-3-(3,4,5-trihydroxyphenyl)acryloylamino]hexyl]-3-(3,4,5-trihydroxyphenyl)acrylamide IC50: 0.006 mM 669796 3.6.5.5 0.0064 - 3-(4-azidophenyl)-2-cyano-N-[3-[2-cyano-3-(3,4-dihydroxyphenyl)acryloylamino]propyl]acrylamide in 10 mM Tris, 10 mM NaCl, 2 mM Mg2+, at 30°C 697337 3.6.5.5 0.0068 - 4-(N,N-dimethyl-N-dodecyl-N-propyl)-4-aza-10-oxa-6-ethyltricyclo[5.2.1]decane-3,5-dione methanesulfonate - 689237 3.6.5.5 0.0071 - (5Z)-5-[4-[3-(dimethylamino)propoxy]benzylidene]-3-ethyl-2-thioxo-1,3-thiazolidin-4-one pH and temperature not specified in the publication 718468 3.6.5.5 0.0073 - sertraline in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C 696551 3.6.5.5 0.0074 - (5Z)-3-benzyl-5-[(6,8-dichloro-4-oxo-4H-chromen-3-yl)methylidene]-2-thioxo-1,3-thiazolidin-4-one pH and temperature not specified in the publication 718468 3.6.5.5 0.0074 - (5Z)-5-(2,1,3-benzoxadiazol-5-ylmethylidene)-2-thioxo-1,3-thiazolidin-4-one pH and temperature not specified in the publication 718468 3.6.5.5 0.0075 - (5Z)-5-(3,5-dichlorobenzylidene)-2-thioxo-1,3-thiazolidin-4-one pH and temperature not specified in the publication 718468 3.6.5.5 0.008 - 2-cyano-N-[3-[2-cyano-3-(3,4-dihydroxy-5-methoxy-phenyl)acryloylamino]pentyl]-3-(3,4-dihydroxy-5-methoxyphenyl)acrylamide IC50: 0.008 mM 669796 3.6.5.5 0.008 - 2-cyano-N-[3-[2-cyano-3-(3,4-dihydroxy-5-methoxyphenyl)acryloylamino]butyl]-3-(3,4-dihydroxy-5-methoxyphenyl)acrylamide IC50: 0.008 mM 669796 3.6.5.5 0.0084 - 4-(N,N-dimethyl-N-dodecyl-N-propyl)-4-aza-10-oxatricyclo[5.2.1]decane-3,5-dione bromide - 689237 3.6.5.5 0.0085 - 4-(N,N-dimethyl-N-dodecyl-N-ethyl)-4-aza-10-oxatricyclo[5.2.1]decane-3,5-dione bromide - 689237 3.6.5.5 0.0089 - 4-(N,N-dimethyl-N-dodecyl-N-ethyl)-4-aza-10-oxatricyclo[5.2.1]decane-3,5-dione methanesulfonate - 689237 3.6.5.5 0.009 - 2-cyano-N-[2-[2-cyano-3-(3,4-dihydroxy-4-methoxyphenyl)acryloylamino]ethyl]-3-(3,4-dihydroxy-5-methoxyphenyl) acrylamide IC50: 0.009 mM 669796 3.6.5.5 0.01 - 3-[(5Z)-5-[(6,8-dichloro-4-oxo-4H-chromen-3-yl)methylidene]-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]propanoic acid pH and temperature not specified in the publication 718468 3.6.5.5 0.0106 - 2,5-bis(4-carboxyanilino)-1,4-benzoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.0111 - 2,5-bis(4-hydroxyanilino)-1,4-benzoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.0112 - 4-(N,N-dimethyl-N-dodecyl-N-propyl)-4-aza-10-oxatricyclo[5.2.1]decane-3,5-dione methanesulfonate - 689237 3.6.5.5 0.0118 - 4-(N,N-dimethyl-N-dodecyl-N-propyl)-4-aza-10-oxa-6-methyltricyclo[5.2.1]decane-3,5-dione methanesulfonate - 689237 3.6.5.5 0.0123 - [(5Z)-5-[(5-chloro-1-benzothiophen-3-yl)methylidene]-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]acetic acid pH and temperature not specified in the publication 718468 3.6.5.5 0.0147 - fluvoxamine in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C 696551 3.6.5.5 0.0185 - 4-amino-3-sulfo-N-(4-carboxybenzyl)-1,8-naphthalimide pH 7.4, 37°C 734826 3.6.5.5 0.0191 - 4-amino-3-sulfo-N-(carboxymethyl)-1,8-naphthalimide pH 7.4, 37°C 734826 3.6.5.5 0.0211 - N-methyl-9,10-ethanoanthracene-9(10H)-propanamine in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C 696551 3.6.5.5 0.0215 - 2,5-bis(4-(hydroxymethyl)phenylamino)-1,4-benzoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.022 - (5Z)-3-benzyl-5-[4-[3-(dimethylamino)propoxy]benzylidene]-2-thioxo-1,3-thiazolidin-4-one pH and temperature not specified in the publication 718468 3.6.5.5 0.0224 - 2-(4-hydroxyanilino)-1,4-naphthoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.0234 - (3S-trans)-3-((1,3-benzodioxol-5-yloxy)methyl)-4-(4-fluorophenyl)-piperidine in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C 696551 3.6.5.5 0.0235 - 3-[(5Z)-5-(2H-chromen-3-ylmethylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]propanoic acid pH and temperature not specified in the publication 718468 3.6.5.5 0.0241 - myristyl trimethyl ammonium bromide in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C 696551 3.6.5.5 0.0254 - 2,5-bis(3-carboxyanilino)-1,4-benzoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.029 - (5Z)-5-[(6,8-dichloro-4-oxo-4H-chromen-3-yl)methylidene]-2-thioxo-1,3-thiazolidin-4-one pH and temperature not specified in the publication 718468 3.6.5.5 0.029 - 2,5-bis(4-carboxybenzylamino)-1,4-benzoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.0295 - 2-(4-(hydroxymethyl)anilino)-1,4-naphthoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.0299 - 3-(9-chloro-5,6-dihydrobenzo[b][1]benzazepin-11-yl)-N,N-dimethylpropan-1-amine in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C 696551 3.6.5.5 0.0303 - 2-(3-(hydroxymethyl)anilino)-1,4-naphthoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.031 - (5Z)-5-(3,5-dichlorobenzylidene)-3-(prop-2-en-1-yl)-2-thioxo-1,3-thiazolidin-4-one pH and temperature not specified in the publication 718468 3.6.5.5 0.0334 - N-methyl-3-phenyl-3-[4-(trifluoromethyl)phenoxy]-propan-1-amine in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C 696551 3.6.5.5 0.0369 - 2-cyano-N-[3-[2-cyano-3-(3,4-dihydroxyphenyl)acryloylamino]-propyl] 3-[4-(3-trifluoromethyl-3H-diazirin-3-yl)phenyl]acrylamide in 10 mM Tris, 10 mM NaCl, 2 mM Mg2+, at 30°C 697337 3.6.5.5 0.0372 - 2-[(8-chlorodibenzo[b,f]thiepin-10-yl)oxy]-N,N-dimethylethanamine in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C 696551 3.6.5.5 0.038 - 2-cyano-3-(3,4-dihydroxyphenyl)acrylic acid 2-[2-cyano-3-(3,4-dihydroxyphenyl)acryloyloxy]propyl ester IC50: 0.038 mM 669796 3.6.5.5 0.042 - 2-cyano-3-(3,4-dihydroxyphenyl)acrylic acid 2-[2-cyano-3-(3,4-dihydroxyphenyl)acryloyloxy]ethyl ester IC50: 0.042 mM 669796 3.6.5.5 0.042 - 3-[(5Z)-5-(biphenyl-4-ylmethylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]propanoic acid pH and temperature not specified in the publication 718468 3.6.5.5 0.043 - (5Z)-5-(quinoxalin-2-ylmethylidene)-2-thioxo-1,3-thiazolidin-4-one pH and temperature not specified in the publication 718468 3.6.5.5 0.043 - 4-(N-methyl-N-ethylpiperidine)-4-aza-10-oxatricyclo[5.2.1]decane-3,5-dione methanesulfonate - 689237 3.6.5.5 0.044 - (2E)-2-cyano-N-(3-[[(2E)-2-cyano-3-(3,4-dimethoxyphenyl)prop-2-enoyl]amino]propyl)-3-(3,4-dihydroxyphenyl)prop-2-enamide in 10 mM Tris, 10 mM NaCl, 2 mM Mg2, at 30°C 697337 3.6.5.5 0.0448 - 4-amino-3-sulfo-N-(4-hydroxybenzyl)-1,8-naphthalimide pH 7.4, 37°C 734826 3.6.5.5 0.0472 - 3-(2-chloro-10H-phenothiazin-10-yl)-N,N-dimethyl-propan-1-amine in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C 696551 3.6.5.5 0.048 - 3-[(5Z)-5-[(5-chloro-1-benzothiophen-3-yl)methylidene]-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]propanoic acid pH and temperature not specified in the publication 718468 3.6.5.5 0.05 - (5Z)-3-benzyl-5-(3,5-dichlorobenzylidene)-2-thioxo-1,3-thiazolidin-4-one pH and temperature not specified in the publication 718468 3.6.5.5 0.0502 - 2,5-bis(2-carboxyanilino)-1,4-benzoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.051 - (2E)-2-cyano-N-(3-[[(2E)-2-cyano-3-(4-hydroxyphenyl)prop-2-enoyl]amino]propyl)-3-(3,4-dihydroxyphenyl)prop-2-enamide in 10 mM Tris, 10 mM NaCl, 2 mM Mg2, at 30°C 697337 3.6.5.5 0.053 - (5Z)-5-(2,1,3-benzoxadiazol-5-ylmethylidene)-3-benzyl-2-thioxo-1,3-thiazolidin-4-one pH and temperature not specified in the publication 718468 3.6.5.5 0.0579 - 2,5-bis(3-hydroxyanilino)-1,4-benzoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.061 - 2-cyano-3-(3,4-dihydroxyphenyl)acrylic acid 2-[2-cyano-3-(3,4-dihydroxyphenyl)acryloyloxy]butyl ester IC50: 0.061 mM 669796 3.6.5.5 0.062 - 4-amino-3-sulfo-N-(5-hydroxypentyl)-1,8-naphthalimide pH 7.4, 37°C 734826 3.6.5.5 0.064 - 3-(10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5-ylidene)-N-methyl-1-propanamine in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C 696551 3.6.5.5 0.0703 - 4-amino-3-sulfo-N-benzyl-1,8-naphthalimide pH 7.4, 37°C 734826 3.6.5.5 0.073 - [(5Z)-5-(biphenyl-4-ylmethylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]acetic acid pH and temperature not specified in the publication 718468 3.6.5.5 0.08 - 2-cyano-N-[3-[2-cyano-3-(3,4-dihydroxy-5-methoxy-phenyl)acryloylamino]hexyl]-3-(3,4-dihydroxy-5-methoxyphenyl)acrylamide IC50: 0.08 mM 669796 3.6.5.5 0.088 - 4-amino-3-sulfo-N-(3-aminobenzyl)-1,8-naphthalimide pH 7.4, 37°C 734826 3.6.5.5 0.09 - (5Z)-5-(2H-chromen-3-ylmethylidene)-2-thioxo-1,3-thiazolidin-4-one pH and temperature not specified in the publication 718468 3.6.5.5 0.093 - 4-amino-3-sulfo-N-(3-hydroxypropyl)-1,8-naphthalimide pH 7.4, 37°C 734826 3.6.5.5 0.094 - 4-amino-3-sulfo-N-(2-carboxyethyl)-1,8-naphthalimide pH 7.4, 37°C 734826 3.6.5.5 0.096 - 3-[(5Z)-5-(4-bromobenzylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]propanoic acid pH and temperature not specified in the publication 718468 3.6.5.5 0.1 - (1R,2R)-2-(aminomethyl)-N,N-diethyl-1-phenyl-cyclopropane-1-carboxamide IC50 above 0.1 mM, in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C 696551 3.6.5.5 0.1 - 1,2,3,4,10,14b-hexahydro-2-methyldibenzo[c,f]pyrazino[1,2-a]azepine IC50 above 0.1 mM, in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C 696551 3.6.5.5 0.1 - 1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-1,3-dihydro[2]benzofuran-5-carbonitrile IC50 above 0.1 mM, in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C 696551 3.6.5.5 0.1 - 10,11-dihydro-5-[3-(methylamino)propyl]-5H-dibenz[b,f]azepine IC50 above 0.1 mM, in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C 696551 3.6.5.5 0.1 - 3-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)-N,N-dimethylpropan-1-amine IC50 above 0.1 mM, in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C 696551 3.6.5.5 0.1 - 4-[4-(4-chlorophenyl)-4-hydroxy-1-piperidyl]-1-(4-fluorophenyl)-butan-1-one IC50 above 0.1 mM, in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C 696551 3.6.5.5 0.1 - 5H-dibenz[b,f]azepine-5-carboxamide IC50 above 0.1 mM, in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C 696551 3.6.5.5 0.1 - methyl 2-phenyl-2-(2-piperidyl)acetate IC50 above 0.1 mM, in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C 696551 3.6.5.5 0.1 - N-(2-diethylaminoethyl)-2-methoxy-5-methylsulfonyl-benzamide IC50 above 0.1 mM, in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C 696551 3.6.5.5 0.1 - N-[(1-ethylpyrrolidin-2-yl)methyl]-2-methoxy-5-sulfamoyl-benzamide IC50 above 0.1 mM, in 10 mM Tris-HCl, 10 mM NaCl, 2 mM Mg2+, at 30°C 696551 3.6.5.5 0.109 - 2-(3-hydroxyanilino)-1,4-naphthoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.112 - 2,5-bis(4-hydroxybenzylamino)-1,4-benzoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.113 - 4-amino-3-sulfo-N-(5-hydroxyhexyl)-1,8-naphthalimide pH 7.4, 37°C 734826 3.6.5.5 0.116 - 2,5-bis(3-methoxypropylamino)-1,4-benzoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.123 - 4-amino-3-sulfo-N-(4-aminobenzyl)-1,8-naphthalimide pH 7.4, 37°C 734826 3.6.5.5 0.134 - (5Z)-3-benzyl-5-(4-bromobenzylidene)-2-thioxo-1,3-thiazolidin-4-one pH and temperature not specified in the publication 718468 3.6.5.5 0.146 - (2E)-2-cyano-N-(3-[[(2E)-2-cyano-3-phenylprop-2-enoyl]amino]propyl)-3-(3,4-dihydroxyphenyl)prop-2-enamide in 10 mM Tris, 10 mM NaCl, 2 mM Mg2, at 30°C 697337 3.6.5.5 0.15 - 2-(4-hydroxybenzylamino)-1,4-naphthoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.155 - 4-amino-3-sulfo-N-(2-aminobenzyl)-1,8-naphthalimide pH 7.4, 37°C 734826 3.6.5.5 0.159 - 4-amino-3-sulfo-N-(3-hydroxyphenyl)-1,8-naphthalimide pH 7.4, 37°C 734826 3.6.5.5 0.17 - 2,5-bis(4-methoxybenzylamino)-1,4-benzoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.193 - 4-amino-3-sulfo-N-(2-hydroxyethyl)-1,8-naphthalimide pH 7.4, 37°C 734826 3.6.5.5 0.264 - 2-chloro-4-(2-dimethylaminopropylamine)-6-methylpyrimidine pH and temperature not specified in the publication 757390 3.6.5.5 0.273 - 2,5-bis-(benzylamino)-1,4-benzoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.296 - 4-amino-3-sulfo-N-(4-hydroxyphenyl)-1,8-naphthalimide pH 7.4, 37°C 734826 3.6.5.5 0.3 - 2,5-bis(2-(dimethylamino)ethylamino)-1,4-benzoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.3 - 2,5-bis(2-(hydroxymethyl)anilino)-1,4-benzoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.3 - 2,5-bis(3-methoxyanilino)-1,4-benzoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.3 - 2,5-bis(4-methoxyanilino)-1,4-benzoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.3 - 2,5-bis(hexylamino)-1,4-benzoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.3 - 3-sulfo-N-(2-hydroxyethyl)-1,8-naphthalimide pH 7.4, 37°C 734826 3.6.5.5 0.3 - 4-amino-3-sulfo-N-(2-aminoethyl)-1,8-naphthalimide pH 7.4, 37°C 734826 3.6.5.5 0.3 - 4-amino-3-sulfo-N-phenyl-1,8-naphthalimide pH 7.4, 37°C 734826 3.6.5.5 0.3 - 4-sulfo-N-(2-hydroxyethyl)-1,8-naphthalimide pH 7.4, 37°C 734826 3.6.5.5 0.314 - 2-(2-carboxyanilino)-1,4-naphthoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.327 - N1-(4-chloro-6-methylpyrimidin-2-yl)-N3,N3-dimethylpropane-1,3-diamine pH and temperature not specified in the publication 757390 3.6.5.5 0.387 - 2,5-bis(2-bromoanilino)-1,4-benzoquinone pH and temperature not specified in the publication 733785 3.6.5.5 0.404 - 4-(N,N-dimethyl-N-butyl-N-ethyl)-4-aza-10-oxatricyclo[5.2.1]decane-3,5-dione methanesulfonate - 689237 3.6.5.5 0.5 - (2E,2'E)-N,N'-(2-phenoxypropane-1,3-diyl)bis[2-cyano-3-(3,4-dihydroxyphenyl)prop-2-enamide] IC50 above 0.5 mM, in 10 mM Tris, 10 mM NaCl, 2 mM Mg2, at 30°C 697337 3.6.5.5 0.5 - (2E,2'E)-N,N'-(2-propoxypropane-1,3-diyl)bis[2-cyano-3-(3,4-dihydroxyphenyl)prop-2-enamide] IC50 above 0.5 mM, in 10 mM Tris, 10 mM NaCl, 2 mM Mg2, at 30°C 697337 3.6.5.5 0.5 - 4-azido-N-(2-[2-cyano-3-(3,4-dihydroxyphenyl)acryloylamino]-1-[[2-cyano-3-(3,4-dihydroxyphenyl)acryloylamino]methyl]ethyl)-2,3,5,6-tetrafluorobenzamide IC50 above 0.5 mM, in 10 mM Tris, 10 mM NaCl, 2 mM Mg2+, at 30°C 697337 3.6.5.5 0.5 - N-[2-[[(2E)-2-cyano-3-(3,4-dihydroxyphenyl)prop-2-enoyl]amino]-1-([[(2E)-2-cyano-3-(3,4-dihydroxyphenyl)prop-2-enoyl]amino]methyl)ethyl]benzamide IC50 above 0.5 mM, in 10 mM Tris, 10 mM NaCl, 2 mM Mg2, at 30°C 697337 3.6.5.5 0.509 - 4-amino-3-sulfo-N-(2-(dimethylamino)ethyl)-1,8-naphthalimide pH 7.4, 37°C 734826 3.6.5.5 0.58 - 2,5-bis(3-bromopropylamino)-1,4-benzoquinone pH and temperature not specified in the publication 733785