EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.6.5.5 | 0.5 |
- |
4-azido-N-(2-[2-cyano-3-(3,4-dihydroxyphenyl)acryloylamino]-1-[[2-cyano-3-(3,4-dihydroxyphenyl)acryloylamino]methyl]ethyl)-2,3,5,6-tetrafluorobenzamide |
IC50 above 0.5 mM, in 10 mM Tris, 10 mM NaCl, 2 mM Mg2+, at 30°C |
697337 |
3.6.5.5 | 0.5 |
- |
N-[2-[[(2E)-2-cyano-3-(3,4-dihydroxyphenyl)prop-2-enoyl]amino]-1-([[(2E)-2-cyano-3-(3,4-dihydroxyphenyl)prop-2-enoyl]amino]methyl)ethyl]benzamide |
IC50 above 0.5 mM, in 10 mM Tris, 10 mM NaCl, 2 mM Mg2, at 30°C |
697337 |
3.6.5.5 | 0.509 |
- |
4-amino-3-sulfo-N-(2-(dimethylamino)ethyl)-1,8-naphthalimide |
pH 7.4, 37°C |
734826 |
3.6.5.5 | 0.58 |
- |
2,5-bis(3-bromopropylamino)-1,4-benzoquinone |
pH and temperature not specified in the publication |
733785 |