EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
5.3.3.1 | 0.0016 |
- |
trilostane |
27°C, pH 7.4 |
693887 |
5.3.3.1 | 0.00375 |
- |
4alpha,5alpha-epoxy-testosterone |
27°C, pH 7.4 |
693887 |
5.3.3.1 | -999 |
- |
more |
dissociation constants of inhibitors |
702370 |
5.3.3.1 | -999 |
- |
more |
Ki-values for equilenin and 19-nortestosterone, wild-type enzyme and mutant enzyme D99E |
650004 |
5.3.3.1 | 0.00083 |
- |
trilostane |
mutant M187T, 27°C, pH 7.4 |
693887 |
5.3.3.1 | 0.0028 |
- |
4alpha,5alpha-epoxy-testosterone |
mutant M187T, 27°C, pH 7.4 |
693887 |
5.3.3.1 | 0.00184 |
- |
epostane |
mutant Q105M, isoform 1, 27°C, pH 7.4 |
662371 |
5.3.3.1 | 0.00208 |
- |
trilostane |
mutant Q105M, isoform 1, 27°C, pH 7.4 |
662371 |
5.3.3.1 | 0.00164 |
- |
epostane |
mutant Q105M, isoform 2, 27°C, pH 7.4 |
662371 |
5.3.3.1 | 0.00207 |
- |
trilostane |
mutant Q105M, isoform 2, 27°C, pH 7.4 |
662371 |