EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
5.3.3.1 | 0.0028 |
- |
4alpha,5alpha-epoxy-testosterone |
mutant M187T, 27°C, pH 7.4 |
693887 |
5.3.3.1 | 0.00375 |
- |
4alpha,5alpha-epoxy-testosterone |
27°C, pH 7.4 |
693887 |
5.3.3.1 | 0.0041 |
- |
4alpha,5alpha-epoxy-testosterone |
wild-type, 27°C, pH 7.4 |
693887 |
5.3.3.1 | 0.0043 |
- |
4alpha,5alpha-epoxy-testosterone |
mutant S124T, 27°C, pH 7.4 |
693887 |
5.3.3.1 | 0.00007 |
- |
epostane |
mutant Q240R, isoform 1, 27°C, pH 7.4 |
662371 |
5.3.3.1 | 0.00007 |
- |
epostane |
wild-type, isoform 1, 27°C, pH 7.4 |
662371 |
5.3.3.1 | 0.00021 |
- |
epostane |
mutant R240Q, isoform 2, 27°C, pH 7.4 |
662371 |
5.3.3.1 | 0.00098 |
- |
epostane |
wild-type, isoform 2, 27°C, pH 7.4 |
662371 |
5.3.3.1 | 0.00164 |
- |
epostane |
mutant Q105M, isoform 2, 27°C, pH 7.4 |
662371 |
5.3.3.1 | 0.00184 |
- |
epostane |
mutant Q105M, isoform 1, 27°C, pH 7.4 |
662371 |