EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.5.1.33 | -999 |
- |
more |
all the investigated molecules are assumed to act as full competitive inhibitor and analysed according to the non-tight binding Michaelis-Menten model |
765513 |
1.5.1.33 | -999 |
- |
more |
inhibition kinetics, thermal shift assay |
742445 |
1.5.1.33 | 0.000007 |
- |
1-(3,4-dichlorobenzyl)-7-phenyl-1H-benzimidazol-2-amine |
pH and temperature not specified in the publication |
724770 |
1.5.1.33 | 0.0000111 |
- |
methotrexate |
- |
695556 |
1.5.1.33 | 0.000037 |
- |
methyl 1-[(4-[[(2,4-diaminopteridin-6-yl)methyl](methyl)amino]phenyl)carbonyl]piperidine-4-carboxylate |
- |
689793 |
1.5.1.33 | 0.000039 |
- |
methotrexate |
pH and temperature not specified in the publication |
723852 |
1.5.1.33 | 0.000047 |
- |
1-(3,4-dichlorobenzyl)-7-propoxy-1H-benzimidazol-2-amine |
pH and temperature not specified in the publication |
724770 |
1.5.1.33 | 0.000098 |
- |
7-(benzyloxy)-1-(3,4-dichlorobenzyl)-1H-benzimidazol-2-amine |
pH and temperature not specified in the publication |
724770 |
1.5.1.33 | 0.0001 |
- |
methyl 1-[(4-[[(2,4-diaminopteridin-6-yl)methyl]amino]phenyl)carbonyl]piperidine-4-carboxylate |
- |
689793 |
1.5.1.33 | 0.00011 |
- |
(4S)-4-[[(4-[[(2,4-diaminopteridin-6-yl)methyl](methyl)amino]phenyl)carbonyl]amino]-5-oxohexanoic acid |
- |
689793 |