EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
6.3.4.3 | 0.00004 |
- |
methotrexate |
dhch1-/pXNG4-FTL mutant, FV1 line |
700281 |
6.3.4.3 | 0.00042 |
- |
2,4-diamino-6-benzyl-5-(3-phenylpropyl)-pyrimidine |
dhch1-/pXNG4-FTL mutant, FV1 line |
700281 |
6.3.4.3 | 0.00054 |
- |
2,4-diamino-6-(3,4-dichlorophenoxy)-quinazoline |
dhch1-/pXNG4-FTL mutant, FV1 line |
700281 |
6.3.4.3 | 0.0033 |
- |
(2S)-2-[[4-[(6aR)-3-amino-1,9-dioxo-5,6,6a,7-tetrahydro-4H-imidazol[3,4-f]pteridin-8-yl]benzoyl]amino]pentanedioate |
dhch1-/pXNG4-FTL mutant, FV1 line |
700281 |
6.3.4.3 | 0.0037 |
- |
(2S)-2-[[4-[(6aR)-3-amino-1,9-dioxo-5,6,6a,7-tetrahydro-4H-imidazol[3,4-f]pteridin-8-yl]benzoyl]amino]pentanedioate |
WT/pXNG4-FTL mutant, FV1 line |
700281 |