EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.25.1 | 0.00785 |
- |
N-[(1S)-1-benzyl-2-[[(1S)-1-(furan-2-ylcarbonyl)-3-methylbutyl]amino]-2-oxoethyl]-Na-(tert-butoxycarbonyl)-L-phenylalaninamide |
- |
685565 |
3.4.25.1 | 0.0347 |
- |
KAuBr4 |
- |
685936 |
3.4.25.1 | 0.01 |
- |
N-(tert-butoxycarbonyl)-L-alanyl-N5-[(1R)-1-(dihydroxyboranyl)-3-methylbutyl]-N1-(naphthalen-2-ylmethyl)-L-glutamamide |
above, caspase-like, b1 activity of 20S proteasome, pH not specified in the publication, temperature not specified in the publication |
707667 |
3.4.25.1 | 0.01 |
- |
N-(tert-butoxycarbonyl)-L-alanyl-N6-[(1R)-1-(dihydroxyboranyl)-3-methylbutyl]-N-(naphthalen-2-ylmethyl)-6-oxo-L-lysinamide |
above, caspase-like, b1 activity of 20S proteasome, pH not specified in the publication, temperature not specified in the publication |
707667 |
3.4.25.1 | 0.01 |
- |
N-(tert-butoxycarbonyl)-L-isoleucyl-N5-[(1R)-1-(dihydroxyboranyl)-3-methylbutyl]-N1-(naphthalen-2-ylmethyl)-L-glutamamide |
above, caspase-like, b1 activity of 20S proteasome, pH not specified in the publication, temperature not specified in the publication |
707667 |
3.4.25.1 | 0.01 |
- |
N-(tert-butoxycarbonyl)-L-phenylalanyl-N5-[(1R)-1-(dihydroxyboranyl)-3-methylbutyl]-N1-(naphthalen-2-ylmethyl)-L-glutamamide |
above, caspase-like, b1 activity of 20S proteasome, pH not specified in the publication, temperature not specified in the publication |
707667 |
3.4.25.1 | 0.01 |
- |
N-(tert-butoxycarbonyl)glycyl-N6-[(1R)-1-(dihydroxyboranyl)-3-methylbutyl]-N-(naphthalen-2-ylmethyl)-6-oxo-L-lysinamide |
above, caspase-like, b1 activity of 20S proteasome, pH not specified in the publication, temperature not specified in the publication |
707667 |
3.4.25.1 | 0.01 |
- |
N2-(tert-butoxycarbonyl)-N-[(1R)-1-(dihydroxyboranyl)-3-methylbutyl]-3-[(naphthalen-2-ylmethyl)amino]-3-oxo-D-alaninamide |
above, caspase-like, b1 activity of 20S proteasome, pH not specified in the publication, temperature not specified in the publication |
707667 |
3.4.25.1 | 0.01 |
- |
N2-(tert-butoxycarbonyl)-N5-[(1R)-1-(dihydroxyboranyl)-3-methylbutyl]-N1-(naphthalen-2-ylmethyl)-L-glutamamide |
above, chymotrypsin-like, b5 activity of 20S proteasome, pH not specified in the publication, temperature not specified in the publication |
707667 |
3.4.25.1 | 0.01 |
- |
N-(tert-butoxycarbonyl)-L-alanyl-N5-[(1R)-1-(dihydroxyboranyl)-3-methylbutyl]-N1-(naphthalen-2-ylmethyl)-L-glutamamide |
above, trypsin-like, b1 activity of 20S proteasome, pH not specified in the publication, temperature not specified in the publication |
707667 |