EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.4.2.12 | 0.855 |
- |
(1Z)-N'-(benzoyloxy)-3-(2-oxo-1,3-benzoxazol-3(2H)-yl)propanimidamide |
at pH 7.5 and 37°C |
737247 |
2.4.2.12 | 0.0032 |
- |
(2E)-1-(4-[[2-(4-fluorophenyl)-1,3-thiazol-4-yl]methyl]piperazin-1-yl)-3-(pyridin-3-yl)prop-2-en-1-one |
pH and temperature not specified in the publication |
735765 |
2.4.2.12 | 0.00078 |
- |
(2E)-3-(pyridin-3-yl)-1-[4-[4-(trifluoromethoxy)benzyl]piperazin-1-yl]prop-2-en-1-one |
pH and temperature not specified in the publication |
735765 |
2.4.2.12 | 0.00067 |
- |
(2E)-3-(pyridin-3-yl)-N-[4-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]prop-2-enamide |
pH and temperature not specified in the publication |
735765 |
2.4.2.12 | 0.00002453 |
- |
(2E)-3-(pyridin-3-yl)-N-[6-(3-[[4-(trifluoromethyl)phenyl]sulfamoyl]phenyl)hexyl]prop-2-enamide |
pH and temperature not specified in the publication |
758918 |
2.4.2.12 | 0.00001163 |
- |
(2E)-N-(6-[3-[(2,5-dimethylphenyl)sulfamoyl]phenyl]hexyl)-3-(pyridin-3-yl)prop-2-enamide |
pH and temperature not specified in the publication |
758918 |
2.4.2.12 | 0.00000508 |
- |
(2E)-N-(6-[3-[(2-methylphenyl)sulfamoyl]phenyl]hexyl)-3-(pyridin-3-yl)prop-2-enamide |
pH and temperature not specified in the publication |
758918 |
2.4.2.12 | 0.0000097 |
- |
(2E)-N-(6-[3-[(3-chloro-4-fluorophenyl)sulfamoyl]phenyl]hexyl)-3-(pyridin-3-yl)prop-2-enamide |
pH and temperature not specified in the publication |
758918 |
2.4.2.12 | 0.00001228 |
- |
(2E)-N-(6-[3-[(3-methylphenyl)sulfamoyl]phenyl]hexyl)-3-(pyridin-3-yl)prop-2-enamide |
pH and temperature not specified in the publication |
758918 |
2.4.2.12 | 0.00001075 |
- |
(2E)-N-(6-[3-[(4-chlorophenyl)sulfamoyl]phenyl]hexyl)-3-(pyridin-3-yl)prop-2-enamide |
pH and temperature not specified in the publication |
758918 |