EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
   3.4.21.59 | 0.0000000953 |
- |
6-amidino-2-naphthyl p-guanidinobenzoate dimethane sulfonate |
pH 7.8, 37°C |
653005 |
| 3.4.21.59 | 0.00000062 |
- |
CRA-2059 |
pH 8.0, 25°C, tryptase-beta |
652748 |
| 3.4.21.59 | 0.000001 |
- |
RWJ-56423 |
pH 7.4, 37°C |
652748 |
| 3.4.21.59 | 0.0000012 |
- |
rLDT1 |
pH 7.6, 25°C |
651867 |
| 3.4.21.59 | 0.0000015 |
- |
N-[(1S)-5-amino-1-[[5-(4-[[2-(3-chlorophenyl)ethyl]carbamoyl]benzyl)-1,2,4-oxadiazol-3-yl]carbonyl]pentyl]-3,5-difluorobenzamide |
- |
683237 |
| 3.4.21.59 | 0.0000017 |
- |
N-[(1S)-5-amino-1-[[5-(4-[[2-(3-chlorophenyl)ethyl]carbamoyl]benzyl)-1,2,4-oxadiazol-3-yl]carbonyl]pentyl]-3,4-difluorobenzamide |
- |
683237 |
| 3.4.21.59 | 0.0000017 |
- |
N-[(1S)-5-amino-1-[[5-(4-[[2-(3-chlorophenyl)ethyl]carbamoyl]benzyl)-1,2,4-oxadiazol-3-yl]carbonyl]pentyl]-3-fluorobenzamide |
- |
683237 |
| 3.4.21.59 | 0.0000018 |
- |
benzyl [(1S)-5-amino-1-[[5-(4-[[2-(3-chlorophenyl)ethyl]carbamoyl]benzyl)-1,2,4-oxadiazol-3-yl]carbonyl]pentyl]carbamate |
- |
683237 |
| 3.4.21.59 | 0.0000018 |
- |
N-[(1S)-5-amino-1-[[5-(4-[[2-(3-chlorophenyl)ethyl]carbamoyl]benzyl)-1,2,4-oxadiazol-3-yl]carbonyl]pentyl]-4-fluorobenzamide |
- |
683237 |
| 3.4.21.59 | 0.0000019 |
- |
ethyl [(1S)-5-amino-1-[[5-(4-[[2-(3-chlorophenyl)ethyl]carbamoyl]benzyl)-1,2,4-oxadiazol-3-yl]carbonyl]pentyl]carbamate |
- |
683237 |
