EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference  |
|---|
   3.1.4.39 | 0.00011 |
- |
lysophosphatidic acid |
- |
665628 |
| 3.1.4.39 | 0.00021 |
- |
1-linoleoyl-lysophosphatidic acid |
most potent in the inhibition of lysoPLD activity, based on fluoresecent assay, same order of inhibitory potency among lysophosphatidic acid analogs with different acyl chains in the spectrophotometric assay |
680318 |
| 3.1.4.39 | 0.00021 |
- |
sphingosine-1-phosphate |
SIP, inhibition of lysoPLD activity, fluorometric assay |
680318 |
| 3.1.4.39 | 0.00055 |
- |
1-arachidonoyl-lysophosphatidic acid |
inhibition of lysoPLD activity, based on fluoresecent assay, same order of inhibitory potency among lysophosphatidic acid analogs with different acyl chains in the spectrophotometric assay |
680318 |
| 3.1.4.39 | 0.0012 |
- |
1-oleoyl-lysophosphatidic acid |
inhibition of lysoPLD activity, based on fluoresecent assay, same order of inhibitory potency among lysophosphatidic acid analogs with different acyl chains in the spectrophotometric assay |
680318 |
| 3.1.4.39 | 0.00141 |
- |
1-palmitoyl-lysophosphatidic acid |
inhibition of lysoPLD activity,size of acyl chain is crucial for the maximal inhibitory action, fluorometric assay |
680318 |
| 3.1.4.39 | 0.0018 |
- |
1-linoleoyl-lysophosphatidic acid |
competitive inhibition, spectrophotometric assay |
680318 |
| 3.1.4.39 | 0.0018 |
- |
sphingosine-1-phosphate |
SIP, inhibition of lysoPLD activity, spectrophotometric assay |
680318 |
| 3.1.4.39 | 0.00209 |
- |
1-stearoyl-lysophosphatidic acid |
inhibition of lysoPLD activity,size of acyl chain is crucial for the maximal inhibitory action, fluorometric assay |
680318 |
| 3.1.4.39 | 0.0034 |
- |
1-arachidonoyl-lysophosphatidic acid |
inhibition of lysoPLD activity, spectrophotometric assay |
680318 |
