EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.7.12.1 | -999 |
- |
more |
inhibition kinetics of tyrosine kinase inhibitors, recombinant His-tagged wild-type and mutant enzymes |
664012 |
2.7.12.1 | 0.000014 |
- |
tyrphostin |
versus ATP, pH 7.5, 30°C, recombinant mutant Y213F |
664012 |
2.7.12.1 | 0.000017 |
- |
genistein |
versus ATP, pH 7.5, 30°C, recombinant mutant Y213F |
664012 |
2.7.12.1 | 0.000018 |
- |
tyrphostin |
versus ATP, pH 7.5, 30°C, recombinant wild-type enzyme |
664012 |
2.7.12.1 | 0.00002 |
- |
genistein |
versus ATP, pH 7.5, 30°C, recombinant wild-type enzyme |
664012 |
2.7.12.1 | 0.0000254 |
- |
midostaurin |
pH 6.8, 22°C |
739790 |
2.7.12.1 | 0.0000284 |
- |
midostaurin |
pH 6.8, 22°C |
739790 |
2.7.12.1 | 0.000055 |
- |
tyrphostin |
versus ATP, pH 7.5, 30°C, recombinant mutant Y317F |
664012 |
2.7.12.1 | 0.000056 |
- |
staurosporine |
pH 7.5, 30°C, recombinant mutant Y213F |
664012 |
2.7.12.1 | 0.000059 |
- |
genistein |
versus ATP, pH 7.5, 30°C, recombinant mutant Y317F |
664012 |