EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.1.3.9 | 0.00096 |
- |
benzaldehyde dibenzylhydrazone |
- |
650557 |
3.1.3.9 | 0.00096 |
- |
tetrahydrothiophene-2-carbaldehyde dibenzylhydrazone |
- |
650557 |
3.1.3.9 | 0.001 |
0.007 |
tungstate |
in detergent treated microsomes |
649729 |
3.1.3.9 | 0.00121 |
- |
4-methoxyphenyl-[4-(4-trifluoromethoxyphenyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-5-yl]methanone |
disrupted microsomes |
650948 |
3.1.3.9 | 0.00128 |
- |
3,4-dichlorobenzaldehyde dibenzylhydrazone |
- |
650557 |
3.1.3.9 | 0.00154 |
- |
4-hydroxybenzaldehyde dibenzylhydrazone |
- |
650557 |
3.1.3.9 | 0.00154 |
- |
4-methoxyphenyl-[4-(4-methoxyphenyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-5-yl]methanone |
disrupted microsomes |
650948 |
3.1.3.9 | 0.0022 |
- |
vanadate |
in detergent treated microsomes |
649729 |
3.1.3.9 | 0.0033 |
- |
4-methoxyphenyl-[4-(4-methoxyphenyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-5-yl]methanone |
intact microsomes |
650948 |
3.1.3.9 | 0.004 |
- |
4-methoxyphenyl-[4-(4-trifluoromethoxyphenyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-5-yl]methanone |
intact microsomes |
650948 |