EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
6.3.4.14 | 0.000005 |
- |
6-(2,6-dibromophenyl)pyrido[2,3-d]pyrimidine-2,7-diamine |
or below, wild-type |
706519 |
6.3.4.14 | 0.000028 |
- |
6-(2,6-dimethoxyphenyl)pyrido[2,3-d]pyrimidine-2,7-diamine |
wild-type |
706519 |
6.3.4.14 | 0.00016 |
- |
6-(2,6-dibromophenyl)pyrido[2,3-d]pyrimidine-2,7-diamine |
mutant H438P |
706519 |
6.3.4.14 | 0.00056 |
- |
6-(2,6-dibromophenyl)pyrido[2,3-d]pyrimidine-2,7-diamine |
mutant I437T |
706519 |
6.3.4.14 | 0.0012 |
- |
6-(2,6-dimethoxyphenyl)pyrido[2,3-d]pyrimidine-2,7-diamine |
wild-type |
706519 |
6.3.4.14 | 0.0073 |
- |
6-(2,6-dimethoxyphenyl)pyrido[2,3-d]pyrimidine-2,7-diamine |
wild-type |
706519 |