EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.22.8 | 0.032 |
- |
diallyl-2,4,4-trimethyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-2-ylphosphonate |
in 100 mM Tris-HCl buffer, pH 7.4, at 37°C |
718180 |
3.4.22.8 | 0.036 |
- |
diallyl-7-benzoyl-2,4,4-trimethyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-2-ylphosphonate |
in 100 mM Tris-HCl buffer, pH 7.4, at 37°C |
718180 |
3.4.22.8 | 0.07 |
- |
dimethyl-7-benzoyl-2,4,4-trimethyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-2-ylphosphonate |
in 100 mM Tris-HCl buffer, pH 7.4, at 37°C |
718180 |
3.4.22.8 | 0.08 |
- |
diethyl-2,4,4,9-tetramethyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-2-ylphosphonate |
in 100 mM Tris-HCl buffer, pH 7.4, at 37°C |
718180 |
3.4.22.8 | 0.09 |
- |
diallyl-7,8-dichloro-2,4,4-trimethyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-2-ylphosphonate |
in 100 mM Tris-HCl buffer, pH 7.4, at 37°C |
718180 |
3.4.22.8 | 0.14 |
- |
dibutyl-7,8-dichloro-2,4,4-trimethyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-2-ylphosphonate |
in 100 mM Tris-HCl buffer, pH 7.4, at 37°C |
718180 |
3.4.22.8 | 0.15 |
- |
diallyl-2,4,4,9-tetramethyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-2-ylphosphonate |
in 100 mM Tris-HCl buffer, pH 7.4, at 37°C |
718180 |
3.4.22.8 | 0.175 |
- |
dibutyl-2,4,4,9-tetramethyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-2-ylphosphonate |
in 100 mM Tris-HCl buffer, pH 7.4, at 37°C |
718180 |
3.4.22.8 | 0.22 |
- |
diethyl-7,8-dichloro-2,4,4-trimethyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-2-ylphosphonate |
in 100 mM Tris-HCl buffer, pH 7.4, at 37°C |
718180 |
3.4.22.8 | 0.278 |
- |
dimethyl-2,4,4-trimethyl-2,3,4,5-tetrahydro-1H-benzo-[b]-[1,4]diazepin-2-ylphosphonate |
in 100 mM Tris-HCl buffer, pH 7.4, at 37°C |
718180 |