EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.2.1.22 | 0.000048 |
- |
1-deoxygalactonojirimycin |
IC50 48 nM with mutant enzyme S65A |
654330 |
3.2.1.22 | 0.000058 |
- |
1-deoxygalactonojirimycin |
IC50 58 nM with mutant enzyme S65D |
654330 |
3.2.1.22 | 0.000059 |
- |
1-deoxygalactonojirimycin |
IC50 59 nM with wild-type enzyme |
654330 |
3.2.1.22 | 0.000063 |
- |
1-deoxygalactonojirimycin |
IC50: 63 nM with mutant enzyme S65T |
654330 |
3.2.1.22 | 6.9 |
- |
(2S,3R,4R,5S)-2-(hydroxymethyl)-5-[(methylamino)methyl]pyrrolidine-3,4-diol |
- |
706048 |
3.2.1.22 | 8.1 |
- |
(2S,3R,4R,5S)-2-[(ethylamino)methyl]-5-(hydroxymethyl)pyrrolidine-3,4-diol |
- |
706048 |