EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.7.1.25 | 0.01 |
- |
4-(3-methoxyphenyl)-5-(phenylmethanesulfonyl)-1H-tetrazol-4-ium |
above, pH 8.0, 37°C, recombinant enzyme |
760013 |
2.7.1.25 | 0.01 |
- |
5-bromo-2-chloro-N-(5-sulfanyl-1,3,4-thiadiazol-2-yl)benzamide |
above, pH 8.0, 37°C, recombinant enzyme |
760013 |
2.7.1.25 | 0.01 |
- |
delamanid |
above, pH 8.0, 37°C, recombinant enzyme |
760013 |
2.7.1.25 | 15.7 |
- |
sulfate |
mutant enzyme T61E, pH and temperature not specified in the publication |
738662 |
2.7.1.25 | 0.00047 |
- |
N,N'-[furan-2,5-diylbis(2-chloro-4,1-phenylene)]diguanidine |
pH 8.0, 37°C, recombinant enzyme |
760013 |
2.7.1.25 | 0.00052 |
- |
8-(4-methyl-3-[3-[([2-methyl-5-[(4,6,8-trisulfonaphthalen-1-yl)carbamoyl]phenyl]carbamoyl)amino]benzamido]benzamido)naphthalene-1,3,5-trisulfonic acid |
pH 8.0, 37°C, recombinant enzyme |
760013 |
2.7.1.25 | 0.00138 |
- |
auranofin |
pH 8.0, 37°C, recombinant enzyme |
760013 |
2.7.1.25 | 0.00203 |
- |
N,N'-[furan-2,5-diylbis(3-chloro-4,1-phenylene)]diguanidine |
pH 8.0, 37°C, recombinant enzyme |
760013 |
2.7.1.25 | 0.00427 |
- |
2-cycloheptyl-4-(4-methoxy-3-[4-[4-(2H-tetrazol-5-yl)phenoxy]butoxy]phenyl)-4a,5,8,8a-tetrahydrophthalazin-1(2H)-one |
pH 8.0, 37°C, recombinant enzyme |
760013 |
2.7.1.25 | 0.00473 |
- |
2-cycloheptyl-5-(4-methoxy-3-[4-[4-(2H-tetrazol-5-yl)phenoxy]butoxy]phenyl)-4,4-dimethyl-2,4-dihydro-3H-pyrazol-3-one |
pH 8.0, 37°C, recombinant enzyme |
760013 |