EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.4.2.4 | 0.085 |
- |
(2,4,5-trioxo-3-phenethyl-imidazolidin-1-yl)ethanoic acid |
pH 7.4, 25°C |
722187 |
2.4.2.4 | 0.044 |
- |
(2R,3R,4S,5R)-9-(3,4-dihydroxy-5-trityloxymethyl-tetrahydrofuran-2-yl)-1,9-dihydropurin-6-one |
pH and temperature not specified in the publication |
759143 |
2.4.2.4 | 0.264 |
- |
(3-benzyl-2,4,5-trioxoimidazolidin-1-yl)acetic acid |
pH and temperature not specified in the publication |
759143 |
2.4.2.4 | 0.0537 |
- |
(E)-1-((2-fluorophenyl)(hydroxyimino)methyl)-5-iodopyrimidine-2,4(1H,3H)-dione |
pH 8.4, 30°C |
759147 |
2.4.2.4 | 0.0156 |
- |
(E)-1-((4-chlorophenyl)(hydroxyimino)methyl)-5-iodopyrimidine-2,4(1H,3H)-dione |
pH 8.4, 30°C |
759147 |
2.4.2.4 | 0.0107 |
- |
(E)-1-((4-ethylphenyl)(hydroxyimino)methyl)-5-iodopyrimidine-2,4(1H,3H)-dione |
pH 8.4, 30°C |
759147 |
2.4.2.4 | 0.0413 |
- |
(E)-1-((4-fluorophenyl)(hydroxyimino)methyl)-5-iodopyrimidine-2,4(1H,3H)-dione |
pH 8.4, 30°C |
759147 |
2.4.2.4 | 0.0334 |
- |
(E)-1-((hydroxyimino)(3-methoxyphenyl)methyl)-5-iodopyrimidine-2,4(1H,3H)-dione |
pH 8.4, 30°C |
759147 |
2.4.2.4 | 0.0252 |
- |
(E)-1-((hydroxyimino)(4-methoxyphenyl)methyl)-5-iodopyrimidine-2,4(1H,3H)-dione |
pH 8.4, 30°C |
759147 |
2.4.2.4 | 0.0225 |
- |
(E)-1-((hydroxyimino)(p-tolyl)methyl)-5-iodopyrimidine-2,4(1H,3H)-dione |
pH 8.4, 30°C |
759147 |