EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.4.1.90 | 0.163 |
- |
1-((2R,3S,4R,5R)-tetrahydro-3,4-dihydroxy-5-(hydroxymethyl)furan-2-yl)-5-(1-methyl-1H-indol-4-yl)pyrimidine-2,4(1H,3H)-dione |
pH and temperature not specified in the publication |
756430 |
2.4.1.90 | 0.207 |
- |
1-((2R,3S,4R,5R)-tetrahydro-3,4-dihydroxy-5-(hydroxymethyl)furan-2-yl)-5-(1H-indol-4-yl)pyrimidine-2,4(1H,3H)-dione |
pH and temperature not specified in the publication |
756430 |
2.4.1.90 | 0.25 |
- |
1-((2R,3S,4R,5R)-tetrahydro-3,4-dihydroxy-5-(hydroxymethyl)furan-2-yl)-5-(1H-indol-6-yl)pyrimidine-2,4(1H,3H)-dione |
pH and temperature not specified in the publication |
756430 |
2.4.1.90 | 0.284 |
- |
2-((5-(1,2,3,4-tetrahydro-1-((2R,3S,4R,5R)-tetrahydro-3,4-dihydroxy-5-(hydroxymethyl)furan-2-yl)-2,4-dioxopyrimidin-5-yl)thiophen-2-yl)methylamino)-3-(1H-indol-3-yl)propanoic acid |
pH and temperature not specified in the publication |
756430 |
2.4.1.90 | 1 |
- |
1-((2R,3S,4R,5R)-tetrahydro-3,4-dihydroxy-5-(hydroxymethyl)furan-2-yl)-5-(1H-indazol-4-yl)pyrimidine-2,4(1H,3H)-dione |
IC50 above 1.0 mM, pH and temperature not specified in the publication |
756430 |
2.4.1.90 | 1 |
- |
1-((2R,3S,4R,5R)-tetrahydro-3,4-dihydroxy-5-(hydroxymethyl)furan-2-yl)-5-(1H-indol-5-yl)pyrimidine-2,4(1H,3H)-dione |
IC50 above 1.0 mM, pH and temperature not specified in the publication |
756430 |
2.4.1.90 | 1 |
- |
1-((2R,3S,4R,5R)-tetrahydro-3,4-dihydroxy-5-(hydroxymethyl)furan-2-yl)-5-(2-(4-methylpiperazin-1-yl)pyridin-4-yl)pyrimidine-2,4(1H,3H)-dione |
IC50 above 1.0 mM, pH and temperature not specified in the publication |
756430 |
2.4.1.90 | 1 |
- |
1-((2R,3S,4R,5R)-tetrahydro-3,4-dihydroxy-5-(hydroxymethyl)furan-2-yl)-5-(isoquinolin-4-yl)pyrimidine-2,4(1H,3H)-dione |
IC50 above 1.0 mM, pH and temperature not specified in the publication |
756430 |
2.4.1.90 | 1 |
- |
1-((2R,3S,4R,5R)-tetrahydro-3,4-dihydroxy-5-(hydroxymethyl)furan-2-yl)-5-(pyridin-3-yl)pyrimidine-2,4(1H,3H)-dione |
IC50 above 1.0 mM, pH and temperature not specified in the publication |
756430 |
2.4.1.90 | 1 |
- |
1-((2R,3S,4R,5R)-tetrahydro-3,4-dihydroxy-5-(hydroxymethyl)furan-2-yl)-5-(pyridin-4-yl)pyrimidine-2,4(1H,3H)-dione |
IC50 above 1.0 mM, pH and temperature not specified in the publication |
756430 |