EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
7.1.1.8 | 0.00004 |
- |
antimycin A |
- |
695915 |
7.1.1.8 | 0.00004 |
- |
Myxothiazol |
- |
695915 |
7.1.1.8 | 0.000012 |
- |
ilicicolin H |
a Qn site inhibitor, a 5-(4-hydroxyphenyl)-alpha-pyridone with a decalin ring system, wild-type enzyme IC50: 12 nM |
674702 |
7.1.1.8 | 0.001 |
- |
3-[(2-bromo-4-fluorophenyl)amino]-5-(6-bromopyridin-3-yl)-5-methyl-1,3-oxazolidine-2,4-dione |
above, pH 7.4, 23°C |
724549 |
7.1.1.8 | 0.001 |
- |
3-[(4-bromophenyl)amino]-5-(6-bromopyridin-3-yl)-5-methyl-1,3-oxazolidine-2,4-dione |
above, pH 7.4, 23°C |
724549 |
7.1.1.8 | 0.001 |
- |
4-[[5-(6-bromopyridin-3-yl)-5-methyl-2,4-dioxo-1,3-oxazolidin-3-yl]amino]benzonitrile |
above, pH 7.4, 23°C |
724549 |
7.1.1.8 | 0.001 |
- |
5-(6-bromopyridin-3-yl)-3-[(2,4-diethylphenyl)amino]-5-methyl-1,3-oxazolidine-2,4-dione |
above, pH 7.4, 23°C |
724549 |
7.1.1.8 | 0.001 |
- |
5-(6-bromopyridin-3-yl)-3-[(2,6-diethylphenyl)amino]-5-methyl-1,3-oxazolidine-2,4-dione |
above, pH 7.4, 23°C |
724549 |
7.1.1.8 | 0.001 |
- |
5-(6-bromopyridin-3-yl)-3-[(4-chlorophenyl)amino]-5-methyl-1,3-oxazolidine-2,4-dione |
above, pH 7.4, 23°C |
724549 |
7.1.1.8 | 0.001 |
- |
5-(6-bromopyridin-3-yl)-3-[(4-methoxyphenyl)amino]-5-methyl-1,3-oxazolidine-2,4-dione |
above, pH 7.4, 23°C |
724549 |