EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.22.8 | 0.3 |
- |
dibutyl-2,4,4-trimethyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-2-ylphosphonate |
IC50 above 0.3 mM, in 100 mM Tris-HCl buffer, pH 7.4, at 37°C |
718180 |
3.4.22.8 | 0.3 |
- |
dibutyl-7-benzoyl-2,4,4-trimethyl-2,3,4,5-tetrahydro-1H-benzo-[b][1,4]diazepin-2-ylphosphonate |
IC50 above 0.3 mM, in 100 mM Tris-HCl buffer, pH 7.4, at 37°C |
718180 |
3.4.22.8 | 0.3 |
- |
diethyl-7-benzoyl-2,4,4-trimethyl-2,3,4,5-tetrahydro-1H-benzo-[b][1,4]diazepin-2-ylphosphonate |
IC50 above 0.3 mM, in 100 mM Tris-HCl buffer, pH 7.4, at 37°C |
718180 |
3.4.22.8 | 0.3 |
- |
dimethyl-2,4,4-trimethyl-8-nitro-2,3,4,5-tetrahydro-1H-benzo-[b][1,4]diazepin-2-ylphosphonate |
IC50 above 0.3 mM, in 100 mM Tris-HCl buffer, pH 7.4, at 37°C |
718180 |
3.4.22.8 | 0.49 |
- |
diethyl-2,4,4-trimethyl-8-nitro-2,3,4,5-tetrahydro-1H-benzo-[b][1,4]diazepin-2-ylphosphonate |
in 100 mM Tris-HCl buffer, pH 7.4, at 37°C |
718180 |
3.4.22.8 | 0.78 |
- |
dimethyl-7,8-dichloro-2,4,4-trimethyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-2-ylphosphonate |
in 100 mM Tris-HCl buffer, pH 7.4, at 37°C |
718180 |