EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.24.34 | 0.0081 |
- |
(2R,S)-HONH-Mal(Me/Bn)-1,2,9,10-tetrahydroisoquinolide |
pH 7.6, 25°C |
652712 |
3.4.24.34 | 0.045 |
- |
(2R,S)-HONH-Mal(Me/Bn)-alpha-naphthylamide |
pH 7.6, 25°C |
652712 |
3.4.24.34 | 0.0096 |
- |
(2R,S)-HONH-Mal(Me/Bn)-NH-CH2CH2-Ph |
pH 7.6, 25°C |
652712 |
3.4.24.34 | 0.00024 |
- |
(2R,S)-HONH-Mal(Me/Bn)-NH-CH2CH2CH2-Ph |
pH 7.6, 25°C |
652712 |
3.4.24.34 | 0.00038 |
- |
(2R,S)-HONH-Mal(Me/Bn)-NH-CH2CH2CH2CH2-Ph |
pH 7.6, 25°C |
652712 |
3.4.24.34 | 0.0011 |
- |
(2R,S)-HONH-Mal(Me/Bn)-NHBn |
pH 7.6, 25°C |
652712 |
3.4.24.34 | 0.041 |
- |
(2R,S)-HONH-Mal(Me/Bn)-NHBn-(p-COOH) |
pH 7.6, 25°C |
652712 |
3.4.24.34 | 0.044 |
- |
(2R,S)-HONH-Mal(Me/Bn)-NHPh |
pH 7.6, 25°C |
652712 |
3.4.24.34 | 0.011 |
- |
(2R,S)-HONH-Mal(Me/Bn)-Oet |
pH 7.6, 25°C |
652712 |
3.4.24.34 | 0.041 |
- |
(2R,S)-HONH-Mal(Me/i-Bu)-Oet |
pH 7.6, 25°C |
652712 |