EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.7.4.9 | 1 |
- |
deoxyuridine |
- |
706485 |
2.7.4.9 | 1.02 |
- |
2'-deoxyuridine |
- |
662987 |
2.7.4.9 | 1.04 |
- |
3'-(azidomethyl)-3'-deoxythymidine |
- |
662597 |
2.7.4.9 | 1.1 |
- |
1-[(4aR,5S,7R,7aR)-5-(hydroxymethyl)-2-oxohexahydro-2H-furo[3,4-e][1,3]oxazin-7-yl]-5-methylpyrimidine-2,4(1H,3H)-dione |
- |
662597 |
2.7.4.9 | 1.14 |
- |
2'-deoxy-5-ethyluridine |
- |
662987 |
2.7.4.9 | 1.54 |
- |
1-[(1R,2S,3R,4R)-2,3-dihydroxy-4-(hydroxymethyl)cyclopentyl]-5-methylpyrimidine-2,4(1H,3H)-dione |
with dGMP as substrate, in Tris-HCl (50 mM, pH 7.2), phosphoenolpyruvate (0.5 mM), KCl (40 mM), MgCl2 (2 mM), at 30°C |
723332 |
2.7.4.9 | 2.5 |
- |
1-[(1R,2R,3S,4R)-2,3-dihydroxy-4-(hydroxymethyl)cyclopentyl]-5-methylpyrimidine-2,4(1H,3H)-dione |
with TMP as substrate, in Tris-HCl (50 mM, pH 7.2), phosphoenolpyruvate (0.5 mM), KCl (40 mM), MgCl2 (2 mM), at 30°C |
723332 |