EC Number |
Turnover Number Minimum [1/s] |
Turnover Number Maximum [1/s] |
Substrate |
Reference |
---|
1.1.1.141 | 6.1 |
- |
prostaglandin E2 |
pH 8.0, 25°C, 20 nM [1-(3-methylphenyl)-1H-benzimidazol-5-yl](piperidin-1-yl)methanone |
726267 |
1.1.1.141 | 7.5 |
- |
prostaglandin E2 |
pH 8.0, 25°C, 10 nM 3-(2,5-dimethyl-1-phenyl-1H-pyrrol-3-yl)-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepine |
726267 |
1.1.1.141 | 10.3 |
- |
prostaglandin E2 |
pH 8.0, 25°C, 10 nM [1-(3-methylphenyl)-1H-benzimidazol-5-yl](piperidin-1-yl)methanone |
726267 |
1.1.1.141 | 11.1 |
- |
prostaglandin E2 |
pH 8.0, 25°C, 4 nM 3-(2,5-dimethyl-1-phenyl-1H-pyrrol-3-yl)-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepine |
726267 |
1.1.1.141 | 12.4 |
- |
prostaglandin E2 |
pH 8.0, 25°C, 10 nM 2-([(6-bromo-4H-imidazo[4,5-b]pyridin-2-yl)sulfanyl]methyl)benzonitrile |
726267 |
1.1.1.141 | 13.6 |
- |
prostaglandin E2 |
pH 8.0, 25°C |
726267 |
1.1.1.141 | 14.1 |
- |
prostaglandin E2 |
pH 8.0, 25°C, 10 nM 2-([(6-bromo-4H-imidazo[4,5-b]pyridin-2-yl)sulfanyl]methyl)benzonitrile |
726267 |
1.1.1.141 | 35 |
- |
NAD+ |
37°C, pH 7.5, V186K mutant |
654374 |
1.1.1.141 | 37 |
- |
(5Z,13E)-(15S)-11alpha,15-dihydroxy-9-oxoprost-5,13-dienoate |
37°C, pH 7.5, V186K mutant |
654374 |
1.1.1.141 | 42 |
- |
NAD+ |
37°C, pH 7.5, N91D mutant |
654374 |