EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
1.11.2.2 | dityrosine | inhibits MPO-derived dityrosine formation in a dose-dependent manner | Homo sapiens | |
1.11.2.2 | fisetin | - |
Homo sapiens | |
1.11.2.2 | kaempferol | - |
Homo sapiens | |
1.11.2.2 | luteolin | - |
Homo sapiens | |
1.11.2.2 | myricetin | - |
Homo sapiens | |
1.11.2.2 | Q3GA | inhibits MPO-derived dityrosine formation in a dose-dependent manner | Homo sapiens | |
1.11.2.2 | quercetin | potent inhibitor, inhibits MPO-derived dityrosine formation in a dose-dependent manner | Homo sapiens | |
1.11.2.2 | taxifolin | - |
Homo sapiens |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
1.11.2.2 | Homo sapiens | P05164 | - |
- |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|---|---|---|---|
1.11.2.2 | aorta | atherosclerotic aorta | Homo sapiens | - |
1.11.2.2 | HL-60 cell | - |
Homo sapiens | - |
1.11.2.2 | macrophage | - |
Homo sapiens | - |
1.11.2.2 | sputum | - |
Homo sapiens | - |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
1.11.2.2 | quercetin + H2O2 | - |
Homo sapiens | oxidized quercetin + H2O | - |
? | |
1.11.2.2 | tyrosine + H2O2 | - |
Homo sapiens | dityrosine + H2O | - |
? |
EC Number | Synonyms | Comment | Organism |
---|---|---|---|
1.11.2.2 | MPO | - |
Homo sapiens |
1.11.2.2 | myeloperoxidase | - |
Homo sapiens |
EC Number | IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|---|
1.11.2.2 | 0.00127 | - |
- |
Homo sapiens | quercetin | |
1.11.2.2 | 0.00208 | - |
- |
Homo sapiens | kaempferol | |
1.11.2.2 | 0.00387 | - |
- |
Homo sapiens | fisetin | |
1.11.2.2 | 0.00422 | - |
- |
Homo sapiens | luteolin | |
1.11.2.2 | 0.00663 | - |
- |
Homo sapiens | taxifolin |