Cloned (Comment) | Organism |
---|---|
expression of subunit alpha 1 in Saccharomyces cerevisiae together with dog subunit beta1 | Ovis aries |
Protein Variants | Comment | Organism |
---|---|---|
D714A | insensitive to palytoxin | Ovis aries |
D714E | the IC50 of the palytoxin-induced K+ efflux is 4fold higher than in cells expressing the wild-type enzyme | Ovis aries |
D714R | insensitive to palytoxin | Ovis aries |
K691A | insensitive to palytoxin | Ovis aries |
K691D | insensitive to palytoxin | Ovis aries |
K691R | the EC50 of the palytoxin-induced K+ efflux is 7fold higher than in cells expressing the wild-type enzyme | Ovis aries |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
palytoxin | - |
Ovis aries |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Mg2+ | - |
Ovis aries |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Ovis aries | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
kidney | - |
Ovis aries | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
120 | - |
mutant K691A | Ovis aries |
175 | - |
mutant D714A | Ovis aries |
195 | - |
mutant K691R | Ovis aries |
575 | - |
mutant D714E | Ovis aries |
1105 | - |
wild-type | Ovis aries |