Cloned (Comment) | Organism |
---|---|
expressed in Escherichia coli Rosetta 2 (DE3) cells | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
ADP-D-ribose | - |
Homo sapiens | |
Ethacrynic acid | - |
Homo sapiens | |
patulin | most potent inhibitor | Homo sapiens | |
thimerosal | - |
Homo sapiens | |
triclosan | - |
Homo sapiens |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
2''-O-acetyl-ADP-D-ribose + H2O | Homo sapiens | - |
ADP-D-ribose + acetate | - |
? | |
3''-O-acetyl-ADP-D-ribose + H2O | Homo sapiens | - |
ADP-D-ribose + acetate | - |
? | |
[SRPK2 protein]-ADP-D-ribose + H2O | Homo sapiens | - |
[SRPK2 protein] + ADP-D-ribose | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | Q9BQ69 | - |
- |
Purification (Comment) | Organism |
---|---|
HisTrap column chromatography and Superdex 75 gel filtration | Homo sapiens |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
2''-O-acetyl-ADP-D-ribose + H2O | - |
Homo sapiens | ADP-D-ribose + acetate | - |
? | |
3''-O-acetyl-ADP-D-ribose + H2O | - |
Homo sapiens | ADP-D-ribose + acetate | - |
? | |
[SRPK2 protein]-ADP-D-ribose + H2O | - |
Homo sapiens | [SRPK2 protein] + ADP-D-ribose | - |
? |
Synonyms | Comment | Organism |
---|---|---|
MACROD1 | - |
Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.0025 | - |
at pH 7.5 and 25°C | Homo sapiens | patulin | |
0.0052 | - |
at pH 7.5 and 25°C | Homo sapiens | thimerosal | |
0.027 | - |
at pH 7.5 and 25°C | Homo sapiens | Ethacrynic acid | |
0.1 | - |
at pH 7.5 and 25°C | Homo sapiens | triclosan |