Inhibitors | Comment | Organism | Structure |
---|---|---|---|
2-amino-4-(3-benzoylphenyl)thiazole-5-carboxamide | - |
Human immunodeficiency virus 1 | |
2-amino-4-(3-bromo-4-chlorophenyl)thiazole-5-carboxamide | - |
Human immunodeficiency virus 1 | |
2-amino-4-(3-chlorophenyl)thiazole-5-carboxamide | - |
Human immunodeficiency virus 1 | |
2-amino-4-(3-iodophenyl)thiazole-5-carboxamide | - |
Human immunodeficiency virus 1 | |
2-amino-4-(3-phenylphenyl)thiazole-5-carboxamide | - |
Human immunodeficiency virus 1 | |
2-amino-4-phenylthiazole-5-carboxamide | - |
Human immunodeficiency virus 1 | |
3-(2-cyanoacetyl)phenyl diethyl phosphate | - |
Human immunodeficiency virus 1 | |
3-(3-chlorophenyl)-3-oxopropanenitrile | - |
Human immunodeficiency virus 1 | |
3-(3-iodophenyl)-3-oxopropanamide | - |
Human immunodeficiency virus 1 | |
3-benzoyl-3-oxopropanenitrile | - |
Human immunodeficiency virus 1 | |
3-phenyl-3-oxopropanenitrile | - |
Human immunodeficiency virus 1 | |
4-(3-benzoylphenyl)thiazole-5-carboxamide | - |
Human immunodeficiency virus 1 | |
4-(3-bromo-4-chlorophenyl)-1H-imidazole-5-carboxamide | - |
Human immunodeficiency virus 1 | |
4-(3-bromo-4-chlorophenyl)thiazole-5-carboxamide | - |
Human immunodeficiency virus 1 | |
4-(3-chlorophenyl)-1H-imidazole-5-carboxamide | - |
Human immunodeficiency virus 1 | |
4-(3-iodophenyl)-3-oxobutanenitrile | - |
Human immunodeficiency virus 1 | |
4-phenyl-1H-imidazole-5-carboxamide | - |
Human immunodeficiency virus 1 | |
4-phenylthiazole-5-carboxamide | - |
Human immunodeficiency virus 1 | |
nevirapine | - |
Human immunodeficiency virus 1 |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Human immunodeficiency virus 1 | P04585 | - |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
deoxynucleoside triphosphate + DNAn | poly(rA)n¥oligo(dT)12-18 | Human immunodeficiency virus 1 | diphosphate + DNAn+1 | - |
? |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.0017 | - |
- |
Human immunodeficiency virus 1 | nevirapine | |
0.0035 | - |
- |
Human immunodeficiency virus 1 | 4-(3-iodophenyl)-3-oxobutanenitrile | |
0.0041 | - |
- |
Human immunodeficiency virus 1 | 3-(3-chlorophenyl)-3-oxopropanenitrile | |
0.0098 | - |
- |
Human immunodeficiency virus 1 | 3-benzoyl-3-oxopropanenitrile | |
0.0099 | - |
- |
Human immunodeficiency virus 1 | 4-(3-bromo-4-chlorophenyl)-1H-imidazole-5-carboxamide | |
0.0163 | - |
- |
Human immunodeficiency virus 1 | 4-(3-benzoylphenyl)thiazole-5-carboxamide | |
0.0296 | - |
- |
Human immunodeficiency virus 1 | 3-(3-iodophenyl)-3-oxopropanamide | |
0.0334 | - |
- |
Human immunodeficiency virus 1 | 3-phenyl-3-oxopropanenitrile | |
0.0441 | - |
- |
Human immunodeficiency virus 1 | 2-amino-4-(3-benzoylphenyl)thiazole-5-carboxamide | |
0.0544 | - |
- |
Human immunodeficiency virus 1 | 2-amino-4-(3-chlorophenyl)thiazole-5-carboxamide | |
0.0592 | - |
- |
Human immunodeficiency virus 1 | 2-amino-4-(3-phenylphenyl)thiazole-5-carboxamide | |
0.0643 | - |
- |
Human immunodeficiency virus 1 | 3-(2-cyanoacetyl)phenyl diethyl phosphate | |
0.0798 | - |
- |
Human immunodeficiency virus 1 | 4-(3-chlorophenyl)-1H-imidazole-5-carboxamide | |
0.0807 | - |
- |
Human immunodeficiency virus 1 | 2-amino-4-phenylthiazole-5-carboxamide | |
0.0875 | - |
- |
Human immunodeficiency virus 1 | 4-(3-bromo-4-chlorophenyl)thiazole-5-carboxamide | |
0.118 | - |
- |
Human immunodeficiency virus 1 | 2-amino-4-(3-bromo-4-chlorophenyl)thiazole-5-carboxamide | |
0.1254 | - |
- |
Human immunodeficiency virus 1 | 2-amino-4-(3-iodophenyl)thiazole-5-carboxamide | |
0.283 | - |
- |
Human immunodeficiency virus 1 | 4-phenylthiazole-5-carboxamide | |
0.3 | - |
- |
Human immunodeficiency virus 1 | 4-phenyl-1H-imidazole-5-carboxamide |