EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.1.1.21 | -999 |
- |
more |
inhibition kinetics |
738840 |
1.1.1.21 | -999 |
- |
more |
inhibition kinetics and thermodynamic studies of inhibitors binding to the enzyme, overview |
667913 |
1.1.1.21 | -999 |
- |
more |
inhibition kinetics, overview |
722065 |
1.1.1.21 | -999 |
- |
more |
inhibition kinetics, pH dependence of inhibition, overview |
667553 |
1.1.1.21 | 0.000005 |
- |
zopolrestat |
pH 6.2, 30°C, isoform ALR2 |
685547 |
1.1.1.21 | 0.00004 |
- |
(5-chloro-2-[(4-cyanobenzyl)carbamoyl]phenoxy)acetic acid |
mutant T113A/C303D, pH 7.0, 22°C |
685200 |
1.1.1.21 | 0.000043 |
- |
zopolrestat |
pH 6.2, 25°C, recombinant enzyme |
667553 |
1.1.1.21 | 0.00006 |
- |
(5-chloro-2-[(4-cyanobenzyl)carbamoyl]phenoxy)acetic acid |
mutant T113A/C303NpH 7.0, 22°C |
685200 |
1.1.1.21 | 0.000073 |
- |
[5-(4-chlorophenyl)-3-ethyl-1-oxopyrimido[4,5-c]quinolin-2(1H)-yl]acetic acid |
pH 7.5, 25°C |
761030 |
1.1.1.21 | 0.00011 |
- |
(5-chloro-2-[(4-cyanobenzyl)carbamoyl]phenoxy)acetic acid |
mutant T113A, pH 7.0, 22°C |
685200 |