EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
6.3.2.1 | 0.00052 |
- |
N-(4-bromophenyl)-2-methylbenzo[d]imidazo[2,1-b]thiazole-3-carboxamide |
pH 7.8, 37°C, recombinant enzyme |
744489 |
6.3.2.1 | 0.00053 |
- |
2-methyl-N'-(4-phenoxybenzoyl)benzo[d]imidazo[2,1-b]thiazole-3-carbohydrazide |
pH 7.8, 37°C, recombinant enzyme |
744489 |
6.3.2.1 | 0.00058 |
- |
N'-benzylidene-6-methylimidazo[2,1-b]thiazole-5-carbohydrazide |
pH 7.8, 37°C, recombinant enzyme |
744489 |
6.3.2.1 | 0.00064 |
- |
N'-(1-naphthoyl)-6-methylimidazo[2,1-b]thiazole-5-carbohydrazide |
pH 7.8, 37°C, recombinant enzyme |
744489 |
6.3.2.1 | 0.00067 |
- |
6-methyl-N'-(4-(trifluoromethyl)benzylidene)imidazo[2,1-b]thiazole-5-carbohydrazide |
pH 7.8, 37°C, recombinant enzyme |
744489 |
6.3.2.1 | 0.00069 |
- |
N-(4-bromophenyl)-6-methylimidazo[2,1-b]thiazole-5-carboxamide |
pH 7.8, 37°C, recombinant enzyme |
744489 |
6.3.2.1 | 0.00074 |
- |
6-methyl-N-phenylimidazo[2,1-b]thiazole-5-carboxamide |
pH 7.8, 37°C, recombinant enzyme |
744489 |
6.3.2.1 | 0.00084 |
- |
N-benzyl-2-methylbenzo[d]imidazo[2,1-b]thiazole-3-carboxamide |
pH 7.8, 37°C, recombinant enzyme |
744489 |
6.3.2.1 | 0.00102 |
- |
N'-(4-bromobenzylidene)-2-methylbenzo[d]imidazo[2,1-b]thiazole-3-carbohydrazide |
pH 7.8, 37°C, recombinant enzyme |
744489 |
6.3.2.1 | 0.00102 |
- |
N-cyclohexyl-2-methylbenzo[d]imidazo[2,1-b]thiazole-3-carboxamide |
pH 7.8, 37°C, recombinant enzyme |
744489 |