EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
4.3.1.19 | 0.009 |
- |
Ile |
pH 7.5, 30°C, mutant E442A |
729066 |
4.3.1.19 | 0.037 |
- |
Ile |
pH 7.5, 30°C, mutant G350E |
729066 |
4.3.1.19 | 0.067 |
- |
Ile |
pH 7.5, 30°C, wild-type |
729066 |
4.3.1.19 | 0.162 |
- |
Ile |
pH 7.5, 30°C, mutant G445E |
729066 |
4.3.1.19 | 2.32 |
- |
Ile |
pH 7.5, 30°C, mutant F352A |
729066 |
4.3.1.19 | 2.86 |
- |
Ile |
pH 7.5, 30°C, mutant E347F |
729066 |
4.3.1.19 | 3.27 |
- |
Ile |
pH 7.5, 30°C, mutant I460F |
729066 |
4.3.1.19 | 6.99 |
- |
Ile |
pH 7.5, 30°C, mutant R362F |
729066 |