EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.25.1 | -999 |
- |
more |
cell growth inhibition activities, overview |
707667 |
3.4.25.1 | 0.00000865 |
- |
N2-(decylcarbamoyl)-N-[(3E,5S,8S,9E)-2,7-dioxo-5-(propan-2-yl)-1,6-diazacyclododeca-3,9-dien-8-yl]-L-valinamide |
for the chymotrypsin-like activity, pH not specified in the publication, temperature not specified in the publication |
713407 |
3.4.25.1 | 0.0000373 |
- |
MG-132 |
in 10 mM HEPES (pH 7.6), at 37°C |
733663 |
3.4.25.1 | 0.000049 |
- |
glidobactin A |
for the chymotrypsin-like activity, pH not specified in the publication, temperature not specified in the publication |
713407 |
3.4.25.1 | 0.0000796 |
- |
N2-(decylcarbamoyl)-N-[(3E,5S,8S,9E)-2,7-dioxo-5-(propan-2-yl)-1,6-diazacyclododeca-3,9-dien-8-yl]-L-valinamide |
for the trypsin-like activity, pH not specified in the publication, temperature not specified in the publication |
713407 |
3.4.25.1 | 0.000086 |
0.000194 |
(-)-epigallocatechin-3-gallate |
inhibition of the chymotrypsin-like activity of the proteasome in vitro, pH not specified in the publication, temperature not specified in the publication |
702678 |
3.4.25.1 | 0.00022 |
- |
1-[1-(1-[(2,4-dioxoimidazolidin-1-ylimino)-methyl]-2-phenyl-ethylcarbamoyl)-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-(1H-indol) |
pH 7.5, 30°C |
711621 |
3.4.25.1 | 0.00028 |
- |
N-(tert-butoxycarbonyl)glycyl-N5-[(1R)-1-(dihydroxyboranyl)-3-methylbutyl]-N1-(naphthalen-2-ylmethyl)-L-glutamamide |
chymotrypsin-like, b5 activity of 20S proteasome, pH not specified in the publication, temperature not specified in the publication |
707667 |
3.4.25.1 | 0.00054 |
- |
N-(tert-butoxycarbonyl)glycyl-N1-benzyl-N5-[(1R)-1-(dihydroxyboranyl)-3-methylbutyl]-L-glutamamide |
chymotrypsin-like, b5 activity of 20S proteasome, pH not specified in the publication, temperature not specified in the publication |
707667 |
3.4.25.1 | 0.00068 |
- |
N2-(tert-butoxycarbonyl)-N6-[(1R)-1-(dihydroxyboranyl)-3-methylbutyl]-N-(naphthalen-2-ylmethyl)-6-oxo-L-lysinamide |
caspase-like, b1 activity of 20S proteasome, pH not specified in the publication, temperature not specified in the publication |
707667 |