EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.22.60 | 0.0000068 |
- |
(S)-1-(3-fluorobutyl)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin |
- |
696749 |
3.4.22.60 | 0.0000081 |
- |
(S)-1-butyl-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin |
- |
696749 |
3.4.22.60 | 0.000011 |
- |
(S)-1-(4-hydroxybutyl)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin |
- |
696749 |
3.4.22.60 | 0.000011 |
- |
(S)-4-trifluoromethylbenzyl-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin |
- |
696749 |
3.4.22.60 | 0.000028 |
- |
(S)-1-(4-fluorobutyl)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin |
- |
696749 |
3.4.22.60 | 0.000029 |
- |
(S)-4-[5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]-2,3-dioxoindolin-1-yl]butyl 4-methyl-benzenesulfonate |
- |
696749 |
3.4.22.60 | 0.00004 |
- |
(S)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]-1-(3,3,3-trifluoropropyl)isatin |
- |
696749 |
3.4.22.60 | 0.000044 |
- |
(S)-4-fluorobenzyl-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin |
- |
696749 |
3.4.22.60 | 0.000052 |
- |
(S)-1-(3-hydroxypropyl)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin |
- |
696749 |
3.4.22.60 | 0.000058 |
- |
(S)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]-1-propylisatin |
- |
696749 |