EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.22.37 | 0.0000071 |
- |
prodomain of arginine-specific gingipain B |
isoform RgpB, with azocoll as substrate, in 200 mM Tris-HCl, 5 mM CaCl2, 150 mM NaCl, and 0.02% (w/v) NaN3, pH 7.6, supplemented with 10 mM L-cysteine, at 37°C |
731334 |
3.4.22.37 | 0.0000072 |
- |
prodomain of arginine-specific gingipain B |
isoform RgpB, with H-Arg-7-amido-4-methylcoumarin as substrate, in 200 mM Tris-HCl, 5 mM CaCl2, 150 mM NaCl, and 0.02% (w/v) NaN3, pH 7.6, supplemented with 10 mM L-cysteine, at 37°C |
731334 |
3.4.22.37 | 0.0000237 |
- |
prodomain of arginine-specific gingipain B |
isoform RgpB, with Nalpha-benzoyl-L-arginine 4-nitroanilide as substrate, in 200 mM Tris-HCl, 5 mM CaCl2, 150 mM NaCl, and 0.02% (w/v) NaN3, pH 7.6, supplemented with 10 mM L-cysteine, at 37°C |
731334 |
3.4.22.37 | 0.145 |
- |
RRLMAAKAESRK |
at pH 7.5 and 37°C |
731489 |
3.4.22.37 | 0.242 |
- |
RRLMAAKAESR |
at pH 7.5 and 37°C |
731489 |
3.4.22.37 | 0.248 |
- |
RLMAAKAESRK |
at pH 7.5 and 37°C |
731489 |