EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.7.4.21 | 0.0018 |
- |
diphosphoinositol pentakisphosphate |
IC50 for inositol hexakisphosphate kinase activity is 0.0066 mM, IC50 for ATP synthase activity is 0.0018 mM |
642551 |
2.7.4.21 | 0.0018 |
- |
Inositol hexakisphosphate |
IC50 for inositol hexakisphosphate kinase activity is 0.0008 mM, IC50 for ATP synthase activity is 0.0018 mM |
642551 |
2.7.4.21 | 0.00184 |
- |
6-hydroxy-DL-DOPA |
pH 6.95, 37°C |
762234 |
2.7.4.21 | 0.00496 |
- |
myricetin |
pH 6.95, 37°C |
762234 |
2.7.4.21 | 0.0095 |
- |
N2-(m-trifluorobenzyl),N6-(p-nitrobenzyl)purine |
pH 6.95, 37°C, in presence of 0.4 mM 1D-myo-inositol hexakisphosphate |
762234 |
2.7.4.21 | 0.012 |
- |
N2-(m-trifluorobenzyl),N6-(p-nitrobenzyl)purine |
pH 6.95, 37°C |
762234 |
2.7.4.21 | 0.0128 |
- |
1,3,4,5,6-inositol pentakisphosphate |
IC50 for inositol hexakisphosphate kinase activity is 0.022 mM, IC50 for ATP synthase activity is 0.0128 mM |
642551 |
2.7.4.21 | 0.016 |
- |
N2-(m-trifluorobenzyl),N6-(p-nitrobenzyl)purine |
pH 6.95, 37°C, in presence of 0.25 mM ATP |
762234 |
2.7.4.21 | 0.02 |
- |
N2-(m-trifluorobenzyl),N6-(p-nitrobenzyl)purine |
pH 6.95, 37°C, in presence of 0.1 mM 1D-myo-inositol hexakisphosphate |
762234 |
2.7.4.21 | 0.021 |
- |
N2-(m-trifluorobenzyl),N6-(p-nitrobenzyl)purine |
pH 6.95, 37°C, in presence of 0.2 mM 1D-myo-inositol hexakisphosphate |
762234 |