EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.7.11.10 | 0.000005 |
- |
N-[[3-[8-methyl-5-(methylamino)-8H-imidazo[4,5-d]-thiazolo[5,4-b]pyridine-2-yl]phenyl]methyl]methanesulfonamide |
IKK-2 |
705026 |
2.7.11.10 | 0.000006 |
- |
4-methyl-7-methylamino-2-phenyl-4H-imidazo[4,5-d]thiazolo[5,4-b]pyridine |
IKK-2 |
705026 |
2.7.11.10 | 0.000006 |
- |
N,8-dimethyl-2-phenyl-8H-imidazo[4,5-d][1,3]thiazolo[5,4-b]pyridin-5-amine |
- |
702567 |
2.7.11.10 | 0.000007 |
- |
3-[1-methyl-4-(methylamino)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-7-yl]benzonitrile |
- |
702567 |
2.7.11.10 | 0.000007 |
- |
7-(3-fluorophenyl)-N,1-dimethyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-4-amine |
- |
702567 |
2.7.11.10 | 0.000008 |
- |
7-(3-methoxyphenyl)-N,1-dimethyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-4-amine |
- |
702567 |
2.7.11.10 | 0.000009 |
- |
2-methoxy-N-((6-(1-methyl-4-(methylamino)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-7yl)pyridin-2-yl)methyl)acetamide |
IKKbeta catalyzed phosphorylation of IkappaBalpha |
705320 |
2.7.11.10 | 0.00001 |
- |
PHA-408 |
less than 0.000010 |
705312 |
2.7.11.10 | 0.000011 |
- |
4-methyl-7-methylamino-2-phenyl-4H-imidazo[4,5-d]oxazolo[5,4-b]pyridine |
IKK-2 |
705026 |
2.7.11.10 | 0.000011 |
- |
4-[N'-(4,6-dimethylpyrimidin-2-yl)carbamimidamido]-N-(phenylcarbamoyl)benzene-1-sulfonamide |
at 37°C, pH not specified in the publication |
761714 |