EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.4.1.37 | 0.79 |
- |
1-(3-phenyl-1,2,4-thiadiazol-5-yl)piperazine |
pH 6.7, 37°C |
719571 |
2.4.1.37 | 0.97 |
- |
7-aminothieno[2,3-b]pyrazine-6-carboxylic acid |
pH 6.7, 37°C |
719571 |
2.4.1.37 | 1.04 |
- |
1-(3-phenyl-1,2,4-thiadiazol-5-yl)-1,4-diazepane |
pH 6.7, 37°C |
719571 |
2.4.1.37 | 1.2 |
- |
9-D-ribityl-1,3,7-trihydropurine-2,6,8-trione |
pH 7.0, 37°C |
719291 |
2.4.1.37 | 1.28 |
- |
1-(3-methoxyphenyl)piperazine |
pH 6.7, 37°C |
719571 |
2.4.1.37 | 1.56 |
- |
2,3-dimethylquinoxaline-6-carboxylic acid |
pH 6.7, 37°C |
719571 |
2.4.1.37 | 1.61 |
- |
N-methyl-1-[3-(pyridin-4-yl)phenyl]methanamine |
pH 6.7, 37°C |
719571 |
2.4.1.37 | 1.9 |
- |
9-(D-1-deoxy-arabinit-1-yl)-1,3,7-trihydropurine-2,6,8-trione |
pH 7.0, 37°C |
719291 |
2.4.1.37 | 2.11 |
- |
1-(1-benzothiophen-3-yl)methanamine |
pH 6.7, 37°C |
719571 |
2.4.1.37 | 2.16 |
- |
1-methyl-1H-benzotriazole-5-carboxylic acid |
pH 6.7, 37°C |
719571 |