EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.3.1.50 | 0.00000013 |
- |
myriocin |
subunit SPT2, at pH 8.0 and 25°C |
755965 |
2.3.1.50 | 0.00000024 |
- |
[N-[(7S)-4-(3,4-dimethoxybenzoyl)-1-[5-(3-[2-[(3,5-dimethyl-1H-pyrrol-2-yl-kappaN)methylidene]-2H-pyrrol-5-yl-kappaN]propanamido)pentyl]-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-b]pyridin-7-yl]-2-(trifluoromethoxy)benzamidato](difluorido)boron |
subunit SPT2, at pH 8.0 and 25°C |
755965 |
2.3.1.50 | 0.00000041 |
- |
myriocin |
subunit SPT3, at pH 8.0 and 25°C |
755965 |
2.3.1.50 | 0.00000076 |
- |
N-[(7S)-4-(5,6-dimethoxypyridine-3-carbonyl)-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-b]pyridin-7-yl]-2-(trifluoromethoxy)benzamide |
subunit SPT2, at pH 8.0 and 25°C |
755965 |
2.3.1.50 | 0.0000008 |
- |
2-chloro-N-[(7S)-4-(3,4-dimethoxybenzoyl)-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-b]pyridin-7-yl]benzamide |
subunit SPT2, at pH 8.0 and 25°C |
755965 |
2.3.1.50 | 0.0000008 |
- |
[N-[(7S)-4-(3,4-dimethoxybenzoyl)-1-[5-(3-[2-[(3,5-dimethyl-1H-pyrrol-2-yl-kappaN)methylidene]-2H-pyrrol-5-yl-kappaN]propanamido)pentyl]-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-b]pyridin-7-yl]-2-(trifluoromethoxy)benzamidato](difluorido)boron |
subunit SPT3, at pH 8.0 and 25°C |
755965 |
2.3.1.50 | 0.0000016 |
- |
N-[(7S)-4-(5,6-dimethoxypyridine-3-carbonyl)-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-b]pyridin-7-yl]-2-(trifluoromethoxy)benzamide |
subunit SPT3, at pH 8.0 and 25°C |
755965 |
2.3.1.50 | 0.000003 |
- |
sulfamisterin |
antibiotic derived from Pycnidiella sp., IC50: 3 nM |
658109 |
2.3.1.50 | 0.0000032 |
- |
(2S,3R)-2-amino-3,12-dihydroxy-2-hydroxymethyl-octadecanoic acid |
IC50: 3.2 nM |
658109 |
2.3.1.50 | 0.0000035 |
- |
(2S,3R)-2-amino-3-hydroxy-2-hydroxymethyl-12-oxo-octadecanoic acid |
IC50: 3.5 nM |
658109 |