EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.1.1.63 | 0.0000001 |
- |
O6-(4-bromothenyl)guanine |
- |
676204 |
2.1.1.63 | 0.00000093 |
- |
DNA (containing 6-O-methylguanine) |
in 50 mM Tris-HCl pH 8.3, at 37°C |
734793 |
2.1.1.63 | 0.0000014 |
0.000003 |
double-stranded oligonucleotides |
6-O-methylguanine, 6-O-(4-fluorobenzyl)-guanine, 6-O-(3-fluorobenzyl)-guanine, 6-O-(2-fluorobenzyl)-guanine, 6-O-benzylguanine, 6-O-benzylhypoxanthine. IC50: 1.4-3.0 nM |
485491 |
2.1.1.63 | 0.0000018 |
- |
DNA (containing 6-O-carboxymethylguanine) |
in 50 mM Tris-HCl pH 8.3, at 37°C |
734793 |
2.1.1.63 | 0.0000028 |
- |
O6-(4-bromothenyl)-8-thiaguanine |
- |
686337 |
2.1.1.63 | 0.0000034 |
- |
O6-(4-bromothenyl)guanine |
Patrin, PaTrin-2, Lomeguatrib |
686337 |
2.1.1.63 | 0.000006 |
- |
4-[(4-bromothiophen-2-yl)methoxy]-1H-pyrazolo[3,4-d]pyrimidin-6-amine |
- |
686337 |
2.1.1.63 | 0.000018 |
- |
O6-thenylguanine |
- |
686337 |
2.1.1.63 | 0.000022 |
- |
6-(naphtho[1,2-b]thiophen-2-ylmethoxy)-9H-purin-2-amine |
- |
686337 |
2.1.1.63 | 0.000025 |
- |
O4-(4-bromothenylpterin) |
- |
686337 |