EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.1.1.1 | 0.0000068 |
- |
5'-[(3-amino-3-carboxypropyl)[3-(3-carbamoylphenyl)prop-2-yn-1-yl]amino]-5'-deoxyadenosine |
pH 7.5, 37°C |
757404 |
2.1.1.1 | 0.000016 |
- |
5'-[(3-amino-3-carboxypropyl)[3-(3-carbamoyl-4-methylphenyl)prop-2-yn-1-yl]amino]-5'-deoxyadenosine |
pH 7.5, 37°C |
757404 |
2.1.1.1 | 0.000043 |
- |
5'-[[(3S)-3-amino-3-carboxypropyl][4-(3-carbamoylphenyl)butyl]amino]-5'-deoxyadenosine |
pH 7.5, 37°C |
757404 |
2.1.1.1 | 0.000052 |
- |
5'-[(3-amino-3-carboxypropyl)[3-(5-carbamoyl-2-methoxyphenyl)prop-2-yn-1-yl]amino]-5'-deoxyadenosine |
pH 7.5, 37°C |
757404 |
2.1.1.1 | 0.000588 |
- |
6-(methylamino)pyridine-3-carboxamide |
pH 7.5, 37°C |
756192 |
2.1.1.1 | 0.000837 |
- |
6-methoxy-4-methylpyridine-3-carboxamide |
pH 7.5, 37°C |
756192 |
2.1.1.1 | 0.0012 |
- |
3-amino-6-fluoro-1-methylquinolin-1-ium |
pH 8.6, 37°C |
757392 |
2.1.1.1 | 0.0012 |
- |
5-amino-1-methylquinolin-1-ium |
pH 8.6, 37°C |
757392 |
2.1.1.1 | 0.0012 |
- |
S-adenosyl-L-homocysteine |
substrate S-adenosyl-L-methionine, pH 8.6, 37°C |
756053 |
2.1.1.1 | 0.0014 |
- |
5'-deoxy-5'-[[(3S)-3,4-diamino-4-oxobutyl][(naphthalen-2-yl)methyl]amino]adenosine |
pH 8.4, 37°C |
757406 |