EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   1.5.1.33 | 0.00008 |
- |
6-(4-fluorophenyl)-5-phenyl-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine |
pH and temperature not specified in the publication |
743060 |
| 1.5.1.33 | 0.000083 |
- |
6-(4-fluorophenyl)-5-(4-methoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine |
pH and temperature not specified in the publication |
743060 |
| 1.5.1.33 | 0.00009 |
- |
pyrimethamine |
pH 3.7, 22°C |
765513 |
| 1.5.1.33 | 0.00014 |
- |
2-amino-6-phenyl-5-(2-phenylethyl)-3,7-dihydro-4H-pyrrolo[2,3-d]pyrimidin-4-one |
pH and temperature not specified in the publication |
743060 |
| 1.5.1.33 | 0.00015 |
- |
5,6-bis(4-fluorophenyl)-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine |
pH and temperature not specified in the publication |
743060 |
| 1.5.1.33 | 0.000186 |
- |
1-(3,4-dichlorophenyl)-6-(4-nitrophenyl)-1,6-dihydro-1,3,5-triazine-2,4-diamine |
pH 3.7, 22°C, recombinant enzyme |
765513 |
| 1.5.1.33 | 0.00019 |
- |
5,6-bis(4-methylphenyl)-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine |
pH and temperature not specified in the publication |
743060 |
| 1.5.1.33 | 0.00019 |
- |
5-(3-chlorophenyl)-6-(4-fluorophenyl)-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine |
pH and temperature not specified in the publication |
743060 |
| 1.5.1.33 | 0.00025 |
- |
6-(4-bromophenyl)-5-phenyl-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine |
pH and temperature not specified in the publication |
743060 |
| 1.5.1.33 | 0.00041 |
- |
2-amino-5,6-diphenyl-3,7-dihydro-4H-pyrrolo[2,3-d]-pyrimidin-4-one |
pH and temperature not specified in the publication |
743060 |
