EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
1.14.15.16 | 0.000015 |
- |
VID400 |
pH and temperature not specified in the publication |
728214 |
1.14.15.16 | 0.00019 |
- |
1-[4-(1H-imidazol-1-yl)butyl]-4-(3,5-dimethoxystyryl)-1H-indole |
pH 7.5, 37°C |
736056 |
1.14.15.16 | 0.0002 |
- |
1-[4-(1H-imidazol-1-yl)butyl]-4-styryl-1H-indole |
pH 7.5, 37°C |
736056 |
1.14.15.16 | 0.0003 |
- |
N-[2-(1H-imidazol-1-yl)-2-phenylethyl]-4-[(E)-2-phenylethenyl]benzamide |
pH 7.5, 37°C |
736056 |
1.14.15.16 | 0.00036 |
- |
1-[3-(1H-imidazol-1-yl)propyl]-4-styryl-1H-indole |
pH 7.5, 37°C |
736056 |
1.14.15.16 | 0.00044 |
- |
1-[3-(1H-imidazol-1-yl)propyl]-4-(3,5-dimethoxystyryl)-1H-indole |
pH 7.5, 37°C |
736056 |
1.14.15.16 | 0.00047 |
- |
ketoconazole |
pH 7.5, 37°C |
736056 |
1.14.15.16 | 0.00052 |
- |
1-[3-(1H-imidazol-1-yl)propyl]-5-styryl-1H-indole |
pH 7.5, 37°C |
736056 |
1.14.15.16 | 0.00052 |
- |
1-[4-(1H-imidazol-1-yl)butyl]-5-styryl-1H-indole |
pH 7.5, 37°C |
736056 |
1.14.15.16 | 0.0033 |
- |
4-methyl-N-[4-(4-styryl-indol-1-yl)butyl]benzenesulfonamide |
pH 7.5, 37°C |
736056 |