EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
1.14.14.32 | 0.0000012 |
- |
abiraterone |
pH 7.3, 37°C |
727424 |
1.14.14.32 | 0.000012 |
- |
abiraterone |
C17,20-lyase activity, pH 7.3, 37°C |
732996 |
1.14.14.32 | 0.000032 |
- |
ketoconazole |
pH 7.3, 37°C |
727424 |
1.14.14.32 | 0.000039 |
- |
SU10603 |
adrenal cortex microsomes, pH and temperature not specified in the publication |
728827 |
1.14.14.32 | 0.000051 |
- |
ketoconazole |
adrenal cortex microsomes, pH and temperature not specified in the publication |
728827 |
1.14.14.32 | 0.000057 |
- |
1-[7-(4-fluorophenyl)-heptyl]-1H-imidazole |
lyase IC50 value |
693885 |
1.14.14.32 | 0.000058 |
- |
1-[5-(4-bromo-phenyl)-pentyl]-1H-imidazole |
lyase IC50 value |
693885 |
1.14.14.32 | 0.00006 |
- |
3beta-hydroxy-17-(50-[30-methyl]-10,20,40-oxadiazolyl)androst-5,16-diene |
pH 7.3, 37°C |
727424 |
1.14.14.32 | 0.000061 |
- |
SU10603 |
H295R cell assay, pH and temperature not specified in the publication |
728827 |
1.14.14.32 | 0.0000651 |
- |
4-(1H-imidazol-1-ylmethyl)phenyl 4-iodobenzenesulfonate |
at 37°C |
702581 |