EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
1.1.1.64 | 0.000001 |
- |
5-[3,5-dichloro-4-(phosphonoxy)benzylidene]-3-(4-methoxyphenyl)-2-thioxo-1,3-oxazolidin-4-one |
cell-based assay, pH not specified in the publication, temperature not specified in the publication |
724555 |
1.1.1.64 | 0.000002 |
- |
5-(3-bromo-4-hydroxybenzylidene)-3-(4-fluorophenyl)-2-thioxo-1,3-oxazolidin-4-one |
cell-based assay, pH not specified in the publication, temperature not specified in the publication |
724555 |
1.1.1.64 | 0.000002 |
- |
5-(3-bromo-4-hydroxybenzylidene)-3-(4-methylphenyl)-2-thioxo-1,3-oxazolidin-4-one |
cell-based assay, pH not specified in the publication, temperature not specified in the publication |
724555 |
1.1.1.64 | 0.000002 |
- |
5-(3-chloro-5-fluoro-4-hydroxybenzylidene)-3-(4-methoxyphenyl)-2-thioxo-1,3-oxazolidin-4-one |
cell-based assay, pH not specified in the publication, temperature not specified in the publication |
724555 |
1.1.1.64 | 0.000002 |
- |
5-(3-fluoro-4-hydroxybenzylidene)-3-(4-methoxyphenyl)-2-tioxo-1,3-oxazolidin-4-one |
cell-based assay, pH not specified in the publication, temperature not specified in the publication |
724555 |
1.1.1.64 | 0.000006 |
- |
(3alpha,5alpha)-3-[[trans-2,5-dimethyl-4-[[2-(trifluoromethyl)-phenyl]sulfonyl]piperazin-1-yl]methyl]-3-hydroxyandrostan-17-one |
assay uses homogenized cells, pH not specified in the publication, temperature not specified in the publication |
724550 |
1.1.1.64 | 0.000014 |
- |
(3alpha,5alpha)-3-([(2R,5S)-2,5-dimethyl-4-[2-(trifluoromethyl)benzene-1-sulfonyl]piperazin-1-yl]methyl)-3-hydroxyandrostan-17-one |
pH and temperature not specified in the publication |
740143 |
1.1.1.64 | 0.000022 |
- |
(3R,5'S,10S,13S)-5'-benzyl-10,13-dimethyltetradecahydro-6'H-spiro[cyclopenta[a]phenanthrene-3,2'-[1,4]oxazinane]-6',17(2H)-dione |
pH and temperature not specified in the publication |
740143 |
1.1.1.64 | 0.000035 |
0.000057 |
N-Adamantan-1-ylmethyl-N-((3R,10S,13S)-3-hydroxy-10,13-dimethyl-17-oxo-hexadecahydro-cyclopenta[a]phenanthren-3-yl)-butyramide |
IC50: 35-57 nM |
658489 |
1.1.1.64 | 0.000036 |
- |
3-[(4-nitrophenyl)amino]benzoic acid |
pH not specified in the publication, temperature not specified in the publication |
724517 |