EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.7.11.30 | 0.000005 |
0.0195 |
4-phenyl-substituted 5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole derivatives |
IC50 of 0.000005-0.0195 mM |
664318 |
2.7.11.30 | 0.00003 |
0.000555 |
4-phenyl substituted pyrazole inhibitors |
inhibitory potency of 4-phenyl substituted pyrazole derivatives, IC50 of 30-555 nM, overview |
664088 |
2.7.11.30 | 0.000031 |
- |
LY364947 |
IC50 is 31 nM |
664318 |
2.7.11.30 | 0.000034 |
- |
3-((4-(6-methylpyridin-2-yl)-5-(quinolin-6-yl)-1H-imidazol-2-yl)methyl)benzamide |
- |
703244 |
2.7.11.30 | 0.00005 |
0.0013 |
4(quinolin-4-yl)-substituted 5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole derivatives |
IC50 of 0.00005-0.0013 mM |
664318 |
2.7.11.30 | 0.000051 |
- |
LY364947 |
IC50 is 51 nM |
664318 |
2.7.11.30 | 0.00007 |
- |
LY566578 |
competitive to ATP, noncompetitive to the peptide substrate, IC50 is 70 nM, mechanism |
664088 |
2.7.11.30 | 0.00011 |
0.02 |
4-phenyl-substituted 5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole derivatives |
IC50 of 0.00011-0.020 mM, overview |
664318 |
2.7.11.30 | 0.00015 |
0.0051 |
4(quinolin-4-yl)-substituted 5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole derivatives |
IC50 of 0.00015-0.0051 mM, overview |
664318 |
2.7.11.30 | 0.000175 |
- |
LY364947 |
competitive to ATP, noncompetitive to the peptide substrate, IC50 is 175 nM, mechanism |
664088 |