EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
1.1.1.270 | 0.00023 |
- |
trilostane |
IC50: 0.00023 mM |
286478 |
1.1.1.270 | 0.000008 |
- |
(Z)-2-(4-methoxyphenylimino)-7-hydroxy-N-(pyridin-2-yl)-2H-chromene-3-carboxamide |
pH 7.4, 25°C, wild-type enzyme |
724124 |
1.1.1.270 | 0.000043 |
- |
minalrestat |
pH 7.4, 25°C, wild-type enzyme |
724124 |
1.1.1.270 | 0.00006 |
- |
3-(4-hydroxy-2-methoxyphenyl)acrylic acid 3-(3-hydroxyphenyl)propyl ester |
pH 7.4, 25°C, wild-type enzyme |
724124 |
1.1.1.270 | 0.00016 |
- |
Tolrestat |
pH 7.4, 25°C, wild-type enzyme |
724124 |
1.1.1.270 | 0.0004 |
- |
oleanolic acid |
pH 7.4, 25°C, wild-type enzyme |
724124 |
1.1.1.270 | 0.0006 |
- |
bisdemethoxycurcumin |
pH 7.4, 25°C, wild-type enzyme |
724124 |
1.1.1.270 | 0.00086 |
- |
sulindac |
pH 7.4, 25°C, wild-type enzyme |
724124 |
1.1.1.270 | 0.0012 |
- |
zopolrestat |
pH 7.4, 25°C, wild-type enzyme |
724124 |
1.1.1.270 | 0.0015 |
- |
epalrestat |
pH 7.4, 25°C, wild-type enzyme |
724124 |