EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
    2.5.1.21 | 0.0085 |
- |
4-methyl-2-(4'-hydroxybiphenyl)-3,4-dihydro-2H-1,4-benzothiazin-2-ol |
pH and temperature not specified in the publication |
759144 |
| 2.5.1.21 | 0.014 |
- |
4-methyl-2-(4'-trifluromethyl-4-biphenyl)-3,4-dihydro-2H-1,4-benzothiazine-2-ol |
pH and temperature not specified in the publication |
759144 |
| 2.5.1.21 | 0.0153 |
- |
[(1R,5R)-7-chloro-1-(2-methylpropyl)-2-oxo-5-phenyl-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetic acid |
pH and temperature not specified in the publication |
721801 |
| 2.5.1.21 | 0.0176 |
- |
carnosol |
pH 7.4, 37°C |
759842 |
| 2.5.1.21 | 0.0184 |
- |
11,12-di-O-methylcarnosol |
pH 7.4, 37°C |
759842 |
| 2.5.1.21 | 0.02 |
- |
1-[[(1S,5S)-7-chloro-5-(2,3-dimethoxyphenyl)-1-(2-methylpropyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetyl]piperidine-4-carboxylic acid |
pH and temperature not specified in the publication |
721801 |
| 2.5.1.21 | 0.02 |
- |
ethyl [(1R,5S)-7-chloro-5-(2-chlorophenyl)-1-(2-methylpropyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetate |
pH and temperature not specified in the publication |
721801 |
| 2.5.1.21 | 0.02 |
- |
[(1R,5S)-1-benzyl-7-chloro-5-(2-chlorophenyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetic acid |
pH and temperature not specified in the publication |
721801 |
| 2.5.1.21 | 0.02 |
- |
[(1R,5S)-5-(2-chlorophenyl)-1-(2-methylpropyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetic acid |
pH and temperature not specified in the publication |
721801 |
| 2.5.1.21 | 0.02 |
- |
[(1R,5S)-5-(2-chlorophenyl)-7-fluoro-1-(2-methylpropyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetic acid |
pH and temperature not specified in the publication |
721801 |
