EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
7.4.2.8 | 0.016 |
- |
2-[(2-amino-2-oxoethyl)sulfanyl]-N-(2,3-dioxo-1,2,3,4-tetrahydroquinoxalin-6-yl)benzamide |
at pH 8.5 and 25°C |
749486 |
7.4.2.8 | 0.016 |
- |
WEN05-03 |
at pH 8.5 and 25°C |
749486 |
7.4.2.8 | 0.046 |
- |
ethyl [2-(2-[[2-(propan-2-yl)quinazolin-4-yl]sulfanyl]acetamido)-1,3-thiazol-4-yl]acetate |
at pH 8.5 and 25°C |
749486 |
7.4.2.8 | 0.046 |
- |
WEN04-34 |
at pH 8.5 and 25°C |
749486 |
7.4.2.8 | 0.255 |
- |
2-[(2-amino-2-oxoethyl)sulfanyl]-N-[4-(piperidin-1-yl)phenyl]benzamide |
at pH 8.5 and 25°C |
749486 |
7.4.2.8 | 0.44 |
- |
2-[(2-amino-2-oxoethyl)sulfanyl]-N-[1-(cyanomethyl)-2,3-dihydro-1H-indol-7-yl]benzamide |
at pH 8.5 and 25°C |
749486 |
7.4.2.8 | 0.44 |
- |
WEN01-04 |
at pH 8.5 and 25°C |
749486 |
7.4.2.8 | 0.47 |
- |
methyl 4-[2-[(2-amino-2-oxoethyl)sulfanyl]benzamido]-1H-indazole-3-carboxylate |
at pH 8.5 and 25°C |
749486 |
7.4.2.8 | 0.47 |
- |
WEN01-01 |
at pH 8.5 and 25°C |
749486 |
7.4.2.8 | 0.475 |
- |
2-[(2-amino-2-oxoethyl)sulfanyl]-N-(3-oxo-3,4-dihydro-2H-1,4-benzothiazin-6-yl)benzamide |
at pH 8.5 and 25°C |
749486 |