EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
    5.1.1.3 | 0.0002 |
- |
(2R,4S,E)-2-amino-4-(3-phenylprop-2-enyl)pentanedioic acid |
potent competitive inhibitor for RacE2 mutant V149A |
675451 |
| 5.1.1.3 | 0.0002 |
- |
(4R,2S)-2-cinnamyl-4-amino-5-hydroxypentanoic acid |
potent competitive inhibitor for RacE2 mutant V149A |
675451 |
| 5.1.1.3 | 0.0003 |
- |
(2R,4S)-2-amino-4-(2-naphthyl)methyl pentanedioic acid |
potent competitive inhibitor for RacE2 mutant V149A |
675451 |
| 5.1.1.3 | 0.0015 |
- |
(4R,2S)-2-cinnamyl-4-amino-5-hydroxypentanoic acid |
D-glutamate analog, good competitive inhibitor for RacE1 |
675451 |
| 5.1.1.3 | 0.0035 |
- |
(2R,4S,E)-2-amino-4-(3-phenylprop-2-enyl)pentanedioic acid |
D-glutamate analog, good competitive inhibitor for RacE1 |
675451 |
| 5.1.1.3 | 0.0046 |
- |
(2R,4S)-2-amino-4-(2-naphthyl)methyl pentanedioic acid |
D-glutamate analog, good competitive inhibitor for RacE1 |
675451 |
| 5.1.1.3 | 0.0058 |
- |
D-glutamate |
- |
676152 |
| 5.1.1.3 | 0.042 |
- |
2-hydroxy-3,4,5-trioxocyclopent-1-en-1-olate |
pH and temperature not specified in the publication |
713607 |
| 5.1.1.3 | 0.059 |
- |
benzene-1,3-disulfonate |
pH and temperature not specified in the publication |
713607 |
| 5.1.1.3 | 0.064 |
- |
(2R,4S,E)-2-amino-4-(3-phenylprop-2-enyl)pentanedioic acid |
D-glutamate analog, only weak inhibitor of RacE2 |
675451 |
